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Inhibitors of acetylcholinesterase. Crystal structure of neostigmine bromide Trevor J. Petcher and Peter Pauling pp 1 - 2; DOI: 10.1021/jm00283a001 |
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Muscarinic agonists. Crystal and molecular structure of 2-methyl-4-trimethylammoniummethyl-1,3-dioxolane iodide and similar substances Peter Pauling and Trevor J. Petcher pp 3 - 5; DOI: 10.1021/jm00283a002 |
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Solid phase synthesis and antibacterial activity of N-terminal sequences of melittin Linneaus C. Dorman and Lowell D. Markley pp 5 - 9; DOI: 10.1021/jm00283a003 |
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Derivatives of 2-amino-5-nitrothiazole as potential schistosomicides Leslie M. Werbel and Josephine R. Battaglia pp 10 - 16; DOI: 10.1021/jm00283a004 |
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Antimalarials. 5. .alpha.-Dibutylaminomethyl- and .alpha.-(2-piperidyl)-3-quinolinemethanols Robert E. Lutz, Cyrus J. Ohnmacht, and Freddy Davis pp 17 - 24; DOI: 10.1021/jm00283a005 |
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L(S)- and D(R)-3-amino-1-phenylpyrrolidines. Stereoselective antagonists for histamine and acetylcholine receptors in vitro Donald T. Witiak, Zuhair Muhi-Eldeen, Narain Mahishi, O. P. Sethi, and Michael C. Gerald pp 24 - 30; DOI: 10.1021/jm00283a006 |
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Conformational study of .beta.-phenethanolamine receptor sites. 3. Synthesis of the 3-isopropylamino-2-phenyl-trans-2-decalols Edward E. Smissman and Samir El-Antably pp 30 - 32; DOI: 10.1021/jm00283a007 |
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Synthesis of 6-chloro-16-methylene-17.alpha.-hydroxy-21-fluoro-4,6-pregnadiene-3,20-dione 17-acetate, a potent progestational agent Thomas L. Popper, F. E. Carlon, E. L. Shapiro, and R. Neri pp 33 - 35; DOI: 10.1021/jm00283a008 |
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Glyoxalase inhibitors. A possible approach to anticancer agents Robert Vince and Susan Daluge pp 35 - 37; DOI: 10.1021/jm00283a009 |
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Hypocholesterolemic agents. 7. C-17 epimer of 20,25-diazacholesterol Raymond E. Counsell, V. V. Ranade, and Fortune Kohen pp 38 - 40; DOI: 10.1021/jm00283a010 |
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Hypoglycemic cyclic amidines William L. Bencze and L. I. Barsky pp 40 - 44; DOI: 10.1021/jm00283a011 |
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Coenzyme Q. 124. New substituted 2,3-dimethoxy-1,4-benzoquinones as inhibitors of coenzyme Q systems Karl Folkers, Joseph C. Catlin, and G. Doyle Daves pp 45 - 48; DOI: 10.1021/jm00283a012 |
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Depressant 1,2-dihydroquinolines and related derivatives Albert Weissman and James F. Muren pp 49 - 53; DOI: 10.1021/jm00283a013 |
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Synthesis and activity of some 1,2,4-triazolylthiazolidones Miha Tisler, A. Andolsek, Branko Stanovnik, M. Likar, and P. Schauer pp 53 - 54; DOI: 10.1021/jm00283a014 |
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cis-1-[(2-Piperidinocyclohexyl)carbonyl]piperidine and related compounds. Oral hypoglycemic agents Ronald H. Rynbrandt and Fredericka L. Schmidt pp 54 - 56; DOI: 10.1021/jm00283a015 |
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Synthesis of some 10-cycloalkylaminodibenz[b,f]azepines David W. Boykin and Bijan Prasun Das pp 56 - 58; DOI: 10.1021/jm00283a016 |
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Synthesis and chemotherapeutic activity of two metabolites of trimethoprim Arnold Brossi, E. Grunberg, M. Hoffer, and Sidney Teitel pp 58 - 59; DOI: 10.1021/jm00283a017 |
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Preparation and antimicrobial activity of N-thiadiazolylcarbamic acid esters Iradj Lalezari and A. Vahdat pp 59 - 60; DOI: 10.1021/jm00283a018 |
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New series of antiarrhythmic agents. The 2-aminotetralins William Everett Johnson, D. M. Graeff, C. D. St. Dennis, and Arnold R. Martin pp 60 - 62; DOI: 10.1021/jm00283a019 |
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Antimalarial and other biological activities of some 2'-alkyl and 2'-aryl derivatives of cinchona alkaloids John P. Yardley, R. E. Bright, Leo Rane, R. W. Rees, Peter Byrom Russell, and Herchel Smith pp 62 - 65; DOI: 10.1021/jm00283a020 |
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Amine oxide analogs of certain cholinergic agents Joseph G. Cannon, Robert Victor Smith, Glenn A. Fischer, John P. Long, and Frederick W. Benz pp 66 - 68; DOI: 10.1021/jm00283a021 |
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Phenothiazines as local anesthetics Vishweshar N. Sharma, Ramji L. Mital, Sailesh P. Banerjee, and Hoshyari L. Sharma pp 68 - 70; DOI: 10.1021/jm00283a022 |
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Preparation and antimalarial activity of compounds related to dypnone guanylhydrazone William T. Colwell, George W. Chan, J. K. Horner, R. M. Parkhurst, and David W. Henry pp 70 - 72; DOI: 10.1021/jm00283a023 |
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Antispasmodic agents. 1. Syntheses and pharmacological activity of aminoalkyl 3-substituted phenylacetates Tetsuji Kametani, Kazuo Kigasawa, Mineharu Hiiragi, T. Aoyama, and Osamu Kusama pp 72 - 75; DOI: 10.1021/jm00283a024 |
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Inhibition of leucine aminopeptidase by halide complexes of platinum Paul Melius, Robert W. Guthrie, and John E. Teggins pp 75 - 76; DOI: 10.1021/jm00283a025 |
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Pyrrolidine derivatives as antispasmodics John K. Sugden and Mohinder Singh pp 76 - 78; DOI: 10.1021/jm00283a026 |
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2,2'-Dialkoxybenzhydrylamides and 2,2'-dialkylbenzhydryl esters of N,N-disubstituted .alpha.-amino acids. Synthesis and pharmacological evaluation Jorge R. Barrio, Armando Novelli, Vicente Ferrari, and Oscar Alonso pp 78 - 80; DOI: 10.1021/jm00283a027 |
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Molecular orbital conformation of phenyl choline ether Lemont B. Kier and Jack M. George pp 80 - 81; DOI: 10.1021/jm00283a028 |
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Synthesis of an allylic alcohol and chloride in the nortriptyline series William B. Lacefield pp 82 - 82; DOI: 10.1021/jm00283a029 |
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Acylthiazolidines Feriano Banci pp 82 - 83; DOI: 10.1021/jm00283a030 |
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Amides of 2-hydroxy-(or alkoxy-) 3-methoxybenzoic acid Georges Tsatsas and E. Costakis pp 83 - 84; DOI: 10.1021/jm00283a031 |
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Carcinogenic activity of dibenzothiophene analogs of p-dimethylaminoazobenzene Ellis Vincent Brown and Russell Isbrandt pp 84 - 85; DOI: 10.1021/jm00283a032 |
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Heterocycles. 4. Syntheses of benzo[h] quinoline derivatives Toshio Moriwake and Masami Inaba pp 85 - 85; DOI: 10.1021/jm00283a033 |
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Amphetamines and Related Compounds Alfred Burger pp 86 - 86; DOI: 10.1021/jm00283a900 |
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Disinfection Alfred Burger pp 86 - 86; DOI: 10.1021/jm00283a901 |
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The History of Penicillin Production Alfred Burger pp 86 - 86; DOI: 10.1021/jm00283a902 |
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The Pharmacopeia of the United States of America Alfred Burger pp 86 - 86; DOI: 10.1021/jm00283a903 |
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Cestocidal activity of 4-alkoxy-1-naphthamidines against dog and cat tapeworms Robert B. Burrows, C. J. Hatton, William G. Lillis, and George R. Hunt pp 87 - 90; DOI: 10.1021/jm00284a001 |
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Syntheses of halogenated phenanthrene amino alcohols as antimalarials Clarence W. Huffman, James T. Traxler, Leroy Krbechek, Richard R. Riter, and Richard G. Wagner pp 90 - 94; DOI: 10.1021/jm00284a002 |
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Chemotherapeutic nitroheterocycles. 6. Substituted 5-aminomethyl-3-(5-nitro-2-imidazolylmethyleneamino)-2-oxazolidinones Clemens Rufer, Hans J. Kessler, and Eberhard Schroeder pp 94 - 96; DOI: 10.1021/jm00284a003 |
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Synthesis and anthelmintic activity of 4-alkoxy-1-naphthamidines Morton Harfenist, Robert B. Burrows, Richard Baltzly, Elizabeth Pedersen, George R. Hunt, Satloo Gurbaxani, J. E. D. Keeling, and Owen D. Standen pp 97 - 103; DOI: 10.1021/jm00284a004 |
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Mitomycin derivatives. 1. Preparation of mitosane and mitosene compounds and their biological activities Shukuo Kinoshita, Keizo Uzu, Kinichi Nakano, Mikio Shimizu, Toshinaka Takahashi, and Masanao Matsui pp 103 - 109; DOI: 10.1021/jm00284a005 |
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Mitomycin derivatives. 2. Derivatives of decarbamoylmitosane and decarbamoylmitosene Shukuo Kinoshita, Keizo Uzu, Kinichi Nakano, and Toshinaka Takahashi pp 109 - 112; DOI: 10.1021/jm00284a006 |
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Chemistry of cephalosporin antibiotics. 22. Chemistry and biological activity of 3-alkoxymethyl cephalosporins John A. Webber, George William Huffman, R. E. Koehler, Charles Franklin Murphy, Charles W. Ryan, Earle M. Van Heyningen, and Robert T. Vasileff pp 113 - 116; DOI: 10.1021/jm00284a007 |
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New class of semisynthetic penicillins and cephalosporins derived from D-2-(1,4-cyclohexadienyl)glycine Joseph E. Dolfini, Harold E. Applegate, Georges Bach, Harold Basch, Jack Bernstein, Joseph Schwartz, and Frank L. Weisenborn pp 117 - 119; DOI: 10.1021/jm00284a008 |
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Irreversible enzyme inhibitors. 180. Irreversible inhibitors of the C'la component of complement derived from m-(phenoxypropoxy) benzamidine and phenoxyacetamide Bernard Randall Baker and Michael Cory pp 119 - 125; DOI: 10.1021/jm00284a009 |
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Folic acid analogs. Modifications in the benzene-ring region. 1. 2'- and 3'-Azafolic acids Eugene Claude Roberts and Y. Fulmer Shealy pp 125 - 130; DOI: 10.1021/jm00284a010 |
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Choline acetyltransferase inhibitors. Styrylpyridine analogs with nitrogen-atom modifications Chester J. Cavallito, Hye Sook Yun, Michael Louis Edwards, and Francis F. Foldes pp 130 - 133; DOI: 10.1021/jm00284a011 |
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Inhibitors of blood platelet aggregation. 1. Biphenylyloxyalkylamines William B. Lacefield, Roy G. Herrmann, Jack Mills, Wilma M. Mills, and J. D. Frank pp 133 - 135; DOI: 10.1021/jm00284a012 |
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Hypocholesterolemic agents. 8. Synthesis of 25-azadihydrolanosterol and derivatives Raymond E. Counsell, Matthias C. Lu, and Fortune Kohen pp 136 - 138; DOI: 10.1021/jm00284a013 |
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Centrally acting cyclic urea, thiourea, and their N,N'-dialkyl derivatives. Structure-activity correlations Eric J. C. Lien and Mehdi Hussain pp 138 - 144; DOI: 10.1021/jm00284a014 |
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Potential nonequilibrium analgetic receptor inactivators. Synthesis and biological activities of N-acylanileridines Philip S. Portoghese, Vasant G. Telang, Akira E. Takemori, and Goro Hayashi pp 144 - 148; DOI: 10.1021/jm00284a015 |
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Structure-activity relation. 3. Structure-activity study of phenethylamines as substrates of biosynthetic enzymes of sympathetic transmitters Toshio Fujita and Takashi Ban pp 148 - 152; DOI: 10.1021/jm00284a016 |
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Effects of a group of dibenzodiazepines on fatal systemic anaphylaxis in mice, rats, and guinea pigs Margaret E. Greig, Anna J. Gibbons, and Gerald Alan Young pp 153 - 156; DOI: 10.1021/jm00284a017 |
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Analogs of amphetamine. 4. Synthesis of metabolites of 1-(2,5-dimethoxy-4-methylphenyl)-2-aminopropane (DOM) Beng-Thong Ho and L. Wayne Tansey pp 156 - 157; DOI: 10.1021/jm00284a018 |
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Analogs of amphetamine. 5. Excretory metabolites of 1-(2,5-dimethoxy-4-methylphenyl)-2-aminopropane (DOM) in rats Beng-Thong Ho, Vicente Estevez, L. Wayne Tansey, Leo F. Englert, Patrick J. Creaven, and William M. McIsaac pp 158 - 160; DOI: 10.1021/jm00284a019 |
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Substituted 1,1-diphenyl-3-aminoprop-1-enes and 1,1-diphenyl-3-aminopropanes as potential antidepressant agents Roy F. Maisey, Geraint Jones, A. R. Somerville, and Brian A. Whittle pp 161 - 164; DOI: 10.1021/jm00284a020 |
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Synthesis of 3-trifluoromethyl steroids Manfred Ernst Wolff and Abraham F. Pascual pp 164 - 167; DOI: 10.1021/jm00284a021 |
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4-Hydroxycoumarins. Synthesis of the metabolites and some other derivatives of warfarin Walter M. Barker, Mark A. Hermodson, and K. P. Link pp 167 - 169; DOI: 10.1021/jm00284a022 |
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Conformationally rigid neurotransmitters. Acetylcholine analogs in the bicyclo[2.2.2] octane system Wendel Lane Nelson and Raymond S. Wilson pp 169 - 171; DOI: 10.1021/jm00284a023 |
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Antimalarials related to aminopyrocatechol dialkyl ethers. Conformation effects Eugene L. Stogryn pp 171 - 173; DOI: 10.1021/jm00284a024 |
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Aminoacyl derivatives of amino sugar nucleosides Herbert A. Friedman pp 174 - 174; DOI: 10.1021/jm00284a025 |
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Heterocyclic N-carboxamides as anticonvulsants Gianfranco Pala, Arturo Donetti, Antonio Mantegani, and Amedeo Omodei-Sale pp 174 - 175; DOI: 10.1021/jm00284a026 |
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Derivatives of 7-oxabicyclo[2.2.1]heptane-exo-cis-2,3-dicarboxylic acid Samuel J. Dominianni and Ronald L. Young pp 175 - 175; DOI: 10.1021/jm00284a027 |
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Potential antidiabetics. 7. N1-(.beta.-hydroxybenzylmethyl)-3-methyl-4-arylhydrazono-2-pyrazolin-5-ones and N1-(.beta.-hydroxybenzylmethyl)-3-methyl-4-arylazo-5-methyl- or -phenylpyrazoles Hari G. Garg and Chandra Prakash pp 175 - 176; DOI: 10.1021/jm00284a028 |
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Chemical Control of Fibrinolysis-Thrombolysis. Theory and Clinical Applications Alfred Burger pp 177 - 177; DOI: 10.1021/jm00284a900 |
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Radiation Protection and Sensitization. Proceedings of the Second International Symposium on Radiosensitizing Drugs, Rome, 1969 Alfred Burger pp 177 - 177; DOI: 10.1021/jm00284a901 |
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Progress in Biochemical Pharmacology: Synthesis and Use of Labelled Lipids and Sterols Alfred Burger pp 177 - 177; DOI: 10.1021/jm00284a902 |
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Kinin Hormones Alfred Burger pp 177 - 177; DOI: 10.1021/jm00284a903 |
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The Pharacological Basis of Therapeutics Alfred Burger pp 177 - 178; DOI: 10.1021/jm00284a904 |
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Human Schistosomiasis Alfred Burger pp 178 - 178; DOI: 10.1021/jm00284a905 |
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A Handbook of Alkaloids and Alkaloid-Containing Plants Alfred Burger pp 178 - 178; DOI: 10.1021/jm00284a906 |
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Analogs of phenothiazines. 3. Synthesis and potential antidepressant activity of some phenothiazine derivatives and related compounds containing a carbocyclic basic side chain Carl Kaiser, David H. Tedeschi, Philip J. Fowler, Alex M. Pavloff, Bruce M. Lester, and Charles L. Zirkle pp 179 - 186; DOI: 10.1021/jm00285a001 |
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Anticonvulsants. 1. Alkoxymethyl derivatives of barbiturates and diphenylhydantoin Julius A. Vida, Carlos M. Samour, and John F. Reinhard pp 187 - 189; DOI: 10.1021/jm00285a002 |
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Anticonvulsants. 2. Acyloxymethyl and halomethyl derivatives of barbituric acid and diphenylhydantoin Julius A. Vida, William R. Wilber, and John F. Reinhard pp 190 - 193; DOI: 10.1021/jm00285a003 |
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Synthesis and identification of metabolites resulting from the biotransformation of DL-methadone in man and in the rat Albert E. Pohland, Harold E. Boaz, and Hugh Richard Sullivan pp 194 - 197; DOI: 10.1021/jm00285a004 |
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Antimalarials. 6. New .alpha.-alkylaminomethyl-4-quinolinemethanols Robert E. Lutz, Atul R. Patel, Cyrus J. Ohnmacht, D. P. Clifford, and A. S. Crosby pp 198 - 202; DOI: 10.1021/jm00285a005 |
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Biologically oriented organic sulfur chemistry. 7. Carbonyl disulfides as inhibitory agents for Histoplasma capsulatum Lamar Field, Wayne S. Hanley, Ilda McVeigh, and Zoe Evans pp 202 - 206; DOI: 10.1021/jm00285a006 |
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2-Amino-4-hydroxy-6-arylaminoethylpteridines as potential antimalarial agents Joseph I. DeGraw, Vernon H. Brown, M. Cory, Panayotis Tsakotellis, Roy L. Kisliuk, and Yvette Gaumont pp 206 - 210; DOI: 10.1021/jm00285a007 |
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.alpha.-Fluoro- and .alpha.-hydroxypyridylalanines Scotty J. Norton, P. Timothy Sullivan, and Cynthia B. Sullivan pp 211 - 214; DOI: 10.1021/jm00285a008 |
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Quaternary furyl-, thienyl-, and pyrrolylpyridinium salts. Oral hypoglycemic agents Gretchen E. Wiegand, Victor J. Bauer, Sidney R. Safir, D. A. Blickens, and S. J. Riggi pp 214 - 215; DOI: 10.1021/jm00285a009 |
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Biological evaluation in vivo and in vitro of selected 5.alpha.-cholestane-3.beta.,5.alpha.,6.beta.-triol analogs as hypocholesterolemic agents Donald T. Witiak, Roger A. Parker, Douglas R. Brann, Mary E. Dempsey, Mary C. Ritter, William E. Connor, and D. M. Brahmankar pp 216 - 222; DOI: 10.1021/jm00285a010 |
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Agents for alkylating steroid hormone receptors. 2. 16.alpha.-Substituted progesterone derivatives Alan J. Solo and John O. Gardner pp 222 - 225; DOI: 10.1021/jm00285a011 |
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Vitamin B6 derivatives. 13. Synthesis of tetrahydrothiazine derivatives of vitamin B6 and their biological properties Kentaro Okumura, Tatsuo Oda, Kazuhiko Kondo, Ichizo Inoue, Tamotsu Danno, Hirotsune Yamaguchi, and Kenji Masukawa pp 226 - 229; DOI: 10.1021/jm00285a012 |
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Complexation of ammonium salts with phenols Chester J. Cavallito, Arthur W. Pittman, and Helen Lyong White pp 230 - 233; DOI: 10.1021/jm00285a013 |
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Nonspecific inhibition of enzymes by organic contrast media Joseph H. Lang and Elliott C. Lasser pp 233 - 236; DOI: 10.1021/jm00285a014 |
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Synthetic nonenyl acetates as attractants for female melon flies Martin Jacobson, Irving Keiser, Derrell L. Chambers, Doris H. Miyashita, and Charles Harding pp 236 - 239; DOI: 10.1021/jm00285a015 |
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2,3-Diarylphthalimidines Denis M. Bailey, James E. Siggins, and C. George DeGrazia pp 240 - 241; DOI: 10.1021/jm00285a016 |
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Glutarimide antibiotics. Analogs of streptimidone Gert P. Volpp and Harry Dounchis pp 241 - 242; DOI: 10.1021/jm00285a017 |
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1-Substituted-3-phenylacetamido-4-phenyl-2-azetidinones as potential antibacterials Jack N. Wells and O. Reed Tarwater pp 242 - 244; DOI: 10.1021/jm00285a018 |
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Synthetic biologically active polymers. 7. Antibacterial activity of some sulfonamide-formaldehyde copolymers Loraine G. Donaruma and John Razzano pp 244 - 244; DOI: 10.1021/jm00285a019 |
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New thiocarboxamides derivatives with specific gastric antisecretory properties Xavier B. L. Pascaud, Charles Malen, and Bernard Danree pp 244 - 246; DOI: 10.1021/jm00285a020 |
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Antimicrobial compounds. 1. Synthesis and antimicrobial activity of some alkylidene, cycloalkylidene, and arylidene derivatives of 3-hydrazinopyridazine M. Japelj, M. Likar, B. Drinovec, A. Pollak, A. Povse, and P. Jerman pp 246 - 247; DOI: 10.1021/jm00285a021 |
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Benzothiazolines as antituberculous agents P. J. Palmer, R. B. Trigg, and J. V. Warrington pp 248 - 251; DOI: 10.1021/jm00285a022 |
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Antifungal activity of the thiosemicarbazones of some heterocyclic aldehydes David M. Wiles and Tony Suprunchuk pp 252 - 254; DOI: 10.1021/jm00285a023 |
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Potential antitumor agents. Selenoguanosine and related compounds Shih-Hsi Chu pp 254 - 255; DOI: 10.1021/jm00285a024 |
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Amebicides. l-Emetine derivatives Andrea Pedrazzoli, Boris Gradnik, and L. Dall'Asta pp 255 - 256; DOI: 10.1021/jm00285a025 |
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Charge-spatial models. 2. Cis and trans-3- and -4-carboxycyclohexyl phosphates and the carboxylate esters as analogs of 2'-deoxyuridine 5'-phosphate Mathias P. Mertes and Mohammed T. Shipchandler pp 257 - 258; DOI: 10.1021/jm00285a026 |
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Mustards derived from 7-phenylbenz[a]anthracene Frank A. Vingiello, Sayeed D. Saraf, and Roger G. Duranleau pp 258 - 259; DOI: 10.1021/jm00285a027 |
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Synthesis and anticancer activity of cytosine arabinoside 3-N-oxide (ara-C 3-N-oxide) Leroy B. Townsend, Raymond P. Panzica, and Roland K. Robins pp 259 - 260; DOI: 10.1021/jm00285a028 |
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Further studies in substituted 4H-1,2,4-triazoles for possible hypoglycemic activity Chimanlal V. Deliwala, Moses Y. Mhasalkar, Madhusudan H. Shah, S. T. Nikam, and Kodaganallur G. Anantanarayanan pp 260 - 262; DOI: 10.1021/jm00285a029 |
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Benzocycloalka[1,2-c]pyridazones Richard A. Partyka and Henry M. Holava pp 262 - 264; DOI: 10.1021/jm00285a030 |
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Synthesis of alkylsalicylic acids as antimicrobial agents D. Buckley and John Thomas pp 265 - 265; DOI: 10.1021/jm00285a031 |
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Search for potential oral hypoglycemic agents. Hydrindene derivatives A. U. De and B. P. Saha pp 265 - 266; DOI: 10.1021/jm00285a032 |
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Anti-Trichinella spiralis activity of some 1-carbamoyl-3-methyl-2-pyrazoline-4,5-dione 4-arylhydrazones Hari G. Garg pp 266 - 266; DOI: 10.1021/jm00285a033 |
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Modified syntheses of 2,4,5-trihydroxyphenylalanine, 2,4,5-trihydroxyphenethylamine, and analogs Fred G. H. Lee, Donald E. Dickson, and Albert A. Manian pp 266 - 268; DOI: 10.1021/jm00285a034 |
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Electronic representation of the lipophilic parameter .pi. Arthur Cammarata and Kenneth S. Rogers pp 269 - 274; DOI: 10.1021/jm00286a001 |
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Mechanism of antimalarial activity of chloroquine analogs from quantitative structure-activity studies. Free energy related model George E. Bass, Donna R. Hudson, Jane E. Parker, and William P. Purcell pp 275 - 283; DOI: 10.1021/jm00286a002 |
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Antimalarials. 7-Chloro-4-(substituted amino)quinolines Tara Singh, Robert George Stein, John F. Hoops, John H. Biel, Wallace K. Hoya, and Deanna R. Cruz pp 283 - 286; DOI: 10.1021/jm00286a003 |
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Microbiological reduction of 2-methyl-1,2-di-3-pyridyl-1-propanone (metyrapone) Ralph Howe and Ronald Haywood Moore pp 287 - 288; DOI: 10.1021/jm00286a004 |
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Stereochemical studies on medicinal agents. 9. Bicyclic bases. Synthesis and biological activities of epimeric quaternary derivatives of 2-oxa-5-azabicyclo[2.2.1]heptane Philip S. Portoghese and Jeremiah G. Turcotte pp 288 - 291; DOI: 10.1021/jm00286a005 |
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Synthesis of some 6-chloro-3,7-dihydroxy-.DELTA.5-pregnene derivatives Ronald A. Le Mahieu, Alfred Boris, M. Carson, and Richard W. Kierstead pp 291 - 294; DOI: 10.1021/jm00286a006 |
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Crystalline molecular structures of two derivatives of 2.beta.-hydroxytestosterone having an unusual A-ring conformation William L. Duax, Chaim Eger, S. Pokrywiecki, and Yoshio Osawa pp 295 - 300; DOI: 10.1021/jm00286a007 |
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Nitrones. 3. .alpha.-(5-Nitro-2-furyl)-N-hydroxy alkylnitrones and their derivatives Hyun Koo Kim, Ronald E. Bambury, and Hesham K. Yaktin pp 301 - 304; DOI: 10.1021/jm00286a008 |
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Preparation and antitumor properties of analogs and derivatives of mycophenolic acid Derrick Fleet Jones and Stuart D. Mills pp 305 - 311; DOI: 10.1021/jm00286a009 |
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Potential antitumor agents. 11. 9-Anilinoacridines Bruce F. Cain, G. J. Atwell, and Ralph N. Seelye pp 311 - 315; DOI: 10.1021/jm00286a010 |
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Irreversible enzyme inhibitors. 181. Inhibition of brain choline acetyltransferase by derivatives of 4-stilbazole Bernard Randall Baker and Raymond E. Gibson pp 315 - 322; DOI: 10.1021/jm00286a011 |
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Inhibition of phenethanolamine N-methyltransferase by ring-substituted .alpha.-methylphenethylamines (amphetamines) Ray W. Fuller, Jack Mills, and Max M. Marsh pp 322 - 325; DOI: 10.1021/jm00286a012 |
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.beta.-Adrenergic blocking agents. 9. Absolute configuration of propranolol and of a number of related aryloxypropanolamines and arylethanolamines M. Dukes and Leslie Harold Smith pp 326 - 328; DOI: 10.1021/jm00286a013 |
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Antihypertensive agents. Substituted 3-pyrrolemethylamines William J. Hudak, Charles H. Tilford, and Richard E. Lewis pp 328 - 331; DOI: 10.1021/jm00286a014 |
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5,8-Dihydroharman derivatives. Preparation and biological activities William A. Remers, Eugene N. Greenblatt, Leon Ellenbogen, and Martin J. Weiss pp 331 - 335; DOI: 10.1021/jm00286a015 |
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Synthesis of some s-triazoles with potential analgesic and antiinflammatory activities Thomas George, D. V. Mehta, R. Tahilramani, Joy David, and P. K. Talwalker pp 335 - 338; DOI: 10.1021/jm00286a016 |
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Aza analogs of 5-(p-fluorophenyl)salicylic acid Gordon L. Walford, Howard Jones, and Tsung-Ying Shen pp 339 - 344; DOI: 10.1021/jm00286a017 |
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Terminal dicarboximido analogs of S-2-(.omega.-aminoalkylamino(ethyl dihydrogen phosphorothioates and related compounds as potential antiradiation agents. 1. Phthalimides and saccharins Thomas Patrick Johnston, James R. Piper, Carl R. Stringfellow, and Robert Daryl Elliott pp 345 - 350; DOI: 10.1021/jm00286a018 |
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Terminal dicarboximido analogs of S-2-.omega.-aminoalkylamino)ethyl dihydrogen phosphorothioates and related compounds as potential antiradiation agents. 2. Succinimides, glutarimides, and cis-1,2-cyclohexanedicarboximides Thomas Patrick Johnston, James R. Piper, and Carl R. Stringfellow pp 350 - 354; DOI: 10.1021/jm00286a019 |
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Antistaphylococcal and antifibrinolytic activities of .omega.-amino acids and their L-histidine dipeptides Elton Strauss Cook, Akira Fujii, Kinji Tanaka, and Yoshiki Tsuchiya pp 354 - 357; DOI: 10.1021/jm00286a020 |
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New antiulcer agents. 1. Synthesis and biological activities of 1-acyl-2-, -3-, and -4-substituted benzamidopiperidines Tsutomu Irikura and Kazunori Kasuga pp 357 - 361; DOI: 10.1021/jm00286a021 |
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Synthesis and pharmacological activity of dihydrobenzofurans Mathias P. Mertes, Larry J. Powers, and Milos M. Hava pp 361 - 365; DOI: 10.1021/jm00286a022 |
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Nitrones. 5. Vinylogs of .alpha.-(5-nitro-2-heteroaryl)-N-substituted nitrones Hyun Koo Kim and Ronald E. Bambury pp 366 - 367; DOI: 10.1021/jm00286a023 |
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Novel substrate of adenosine deaminase Howard J. Schaeffer, S. Gurwara, Robert Vince, and S. Bittner pp 367 - 369; DOI: 10.1021/jm00286a024 |
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Xanthoquininic acid derivatives Leonard M. Rice, Bhagvandas S. Sheth, Theodore B. Zalucky, and J. W. Wheeler pp 369 - 370; DOI: 10.1021/jm00286a025 |
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Potential psychotomimetics. Bromomethoxyamphetamines Charles F. Barfknecht and David E. Nichols pp 370 - 372; DOI: 10.1021/jm00286a026 |
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Nicotinic acid esters as coronary vasodilators Dilbagh S. Bariana and M. Savic pp 372 - 373; DOI: 10.1021/jm00286a027 |
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Resolution of DL-.alpha.-methylphenylalanine Frederick W. Bollinger pp 373 - 375; DOI: 10.1021/jm00286a028 |
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Substituted .gamma.,.gamma.-pentamethyleneparaconamides Toshio Moriwake and Osamu Simamura pp 375 - 375; DOI: 10.1021/jm00286a029 |
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Synthesis of 2,3,6-trimethoxy-.beta.-phenethylamine Frederick Benington and Richard D. Morin pp 375 - 376; DOI: 10.1021/jm00286a030 |
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Conformational study of catechol amine receptor sites. 5. Syntheses of dl-3-amino-2-(3,4-dihydroxyphenyl)-trans-2-decalol hydrochlorides Edward E. Smissman and Ronald T. Borchardt pp 377 - 382; DOI: 10.1021/jm00287a001 |
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Conformational study of catechol amine receptor sites. 6. Syntheses of dl-3-amino-2-(3,4-dihydroxyphenyl)-trans-2-decalin hydrochlorides Edward E. Smissman and Ronald T. Borchardt pp 383 - 387; DOI: 10.1021/jm00287a002 |
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Biotransformation of the sedative 1-(p-chlorophenyl)-2,2-dimethyl-1,3-propanediol 3-carbamate in humans and five animal species Hans W. Ruelius, Frazer V. Hadley, and Stephen R. Shrader pp 388 - 393; DOI: 10.1021/jm00287a003 |
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Synthesis and alkaline decomposition of 5-alkyl-5-(1-methyl-3-oxobutyl)barbituric and 2-thiobarbituric acid derivatives F. Ivy Carroll and Abraham Philip pp 394 - 396; DOI: 10.1021/jm00287a004 |
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Inhibitors of platelet aggregation. 1. 5,10-Dihydro-3-(phenyl, thienyl, and furyl)thiazolo[3,2-b][2,4]benzodiazepines and related compounds Edward F. Elslager, J. R. McLean, Salvatore C. Perricone, Doris Potoczak, H. Veloso, Donald F. Worth, and R. H. Wheelock pp 397 - 401; DOI: 10.1021/jm00287a005 |
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Inhibition of glyoxalase I by S-substituted glutathiones Robert Vince, Susan Daluge, and Wallace B. Wadd pp 402 - 404; DOI: 10.1021/jm00287a006 |
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3-Alkyltyrosines. Potential antihypertensive agents Nicolas Zenker, Yale H. Caplan, David A. Blake, and Eugene M. Johnson pp 405 - 408; DOI: 10.1021/jm00287a007 |
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Synthesis and biological activity of some 5-(1-adamantyl)pyrimidines. 2 James P. Jonak, Sigmund F. Zakrzewski, and Lawrence H. Mead pp 408 - 411; DOI: 10.1021/jm00287a008 |
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Derivatives of 4-azahomoadamantane. Their synthesis and biological evaluation J. G. Korsloot and V. G. Keizer pp 411 - 415; DOI: 10.1021/jm00287a009 |
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2-(Alkylthio)adenosines, specific coronary vasodilators M. Helen Maguire, Denis M. Nobbs, Rosemarie Einstein, and John C. Middleton pp 415 - 420; DOI: 10.1021/jm00287a010 |
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Chemistry of cephalosporin antibiotics. 23. 2-Methyl- and 2-methylenecephalosporins Ian Glaisby Wright, C. W. Ashbrook, T. Goodson, G. V. Kaiser, and E. M. Van Heyningen pp 420 - 426; DOI: 10.1021/jm00287a011 |
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Chemistry of cephalosporin antibiotics. 24. 2-Thiomethyl- and 2-thiomethylenecephalosporins Gary V. Kaiser, C. W. Ashbrook, T. Goodson, Ian Glaisby Wright, and E. M. Van Heyningen pp 426 - 429; DOI: 10.1021/jm00287a012 |
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Antitumor activity of some quaternary ammonium compounds. Structure-activity relation Fotios M. Plakogiannis, Eric J. C. Lien, and John A. Biles pp 430 - 432; DOI: 10.1021/jm00287a013 |
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Aminobenzoic acid diuretics. 2. 4-Substituted-3-amino-5-sulfamoylbenzoic acid derivatives Peter W. Feit pp 432 - 439; DOI: 10.1021/jm00287a014 |
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Effect of 2-anilinopyridines on protein synthesis Denis M. Bailey, Robert E. Johnson, J. D. Connolly, and R. A. Ferrari pp 439 - 443; DOI: 10.1021/jm00287a015 |
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Synthesis and local anesthetic activity of certain piperazine and ephedrine derivatives A. F. Youssef, A. A. Abou-Ouf, and M. A. Abdel Kader pp 443 - 445; DOI: 10.1021/jm00287a016 |
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Stable, biologically active indoxyl Souheil E. Saheb and Makhluf J. Haddadin pp 445 - 446; DOI: 10.1021/jm00287a017 |
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Minimal statistical data for structure-function correlations Paul N. Craig, Corwin H. Hansch, James W. McFarland, Yvonne C. Martin, William P. Purcell, and Rudolph Zahradnik pp 447 - 447; DOI: 10.1021/jm00287a018 |
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Synthesis and toxicology of 5,7-dibenzyloxycyclopentenone[2,3-c]coumarin. Model compound of aflatoxin B1 Paul F. Parks and Ching Yung Wang pp 447 - 448; DOI: 10.1021/jm00287a019 |
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Synthetic trypanocides. 2. Substituted 5,6-dihydro[c]benzocarbazoles Sem M. Albonico and Jorge Gallo Pecca pp 448 - 449; DOI: 10.1021/jm00287a020 |
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Nitrofuryl heterocyclics. 2 Peter J. Islip and Michael D. Closier pp 449 - 450; DOI: 10.1021/jm00287a021 |
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Antitumor agents. Schiff bases from benzaldehyde nitrogen mustards and 2-phenyl-4-[(3-amino-4-methoxy)phenyl]thiazole Chimanlal V. Deliwala, J. D. Modi, and S. S. Sabnis pp 450 - 451; DOI: 10.1021/jm00287a022 |
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Halogenated acetyl derivatives and their antitumor activity Arthur Sweeny, Ronald H. Goldfarb, Theodora N. Salmon, Gordon Loewengart, Rita Fox, and Andrew Sicignano pp 451 - 452; DOI: 10.1021/jm00287a023 |
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Synthesis and central nervous system effects of some benzothiazinones Ned D. Heindel, Jack R. Reid, and Joseph E. Willis pp 453 - 453; DOI: 10.1021/jm00287a024 |
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Synthesis, alkylation, and oxidation of thieno[3,4-c]- and -[3,2-c]pyrazoles Victor J. Bauer, Richard P. Williams, and S. R. Safir pp 454 - 456; DOI: 10.1021/jm00287a025 |
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Synthesis and biological study of a series of S-substituted .alpha.-mercaptohippuramides and nitriles Roger Ketcham, Vinod P. Shah, and Grace Lam pp 456 - 458; DOI: 10.1021/jm00287a026 |
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Mannich derivatives of medicinals. 2. Derivatives of some carbonic anhydrase inhibitors George M. Sieger, William C. Barringer, and James E. Krueger pp 458 - 460; DOI: 10.1021/jm00287a027 |
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Synthetic biologically active polymers. 8. Antibacterial activity of some sulfonamide-dimethylolurea copolymers Lorraine G. Donaruma and John R. Dombroski pp 460 - 461; DOI: 10.1021/jm00287a028 |
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Improved synthesis of diaveridine, trimethoprim, and closely related 2,4-diaminopyrimidines Arnold Brossi, Max Hoffer, Emanuel Grunberg, and Milan Mitrovic pp 462 - 463; DOI: 10.1021/jm00287a029 |
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Seeds as sources of L-Dopa Melvin E. Daxenbichler, Cecil H. VanEtten, E. Ann Hallinan, Fontaine R. Earle, and Arthur S. Barclay pp 463 - 465; DOI: 10.1021/jm00287a030 |
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2(5-Nitro-2-thienyl)cinchoninic acids Iradj Lalezari, F. Ghabgharan, and R. Maghsoudi pp 465 - 465; DOI: 10.1021/jm00287a031 |
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Analogs of albizziin Charles G. Skinner and Dale R. Sargent pp 465 - 466; DOI: 10.1021/jm00287a032 |
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Conversion of ergosterol into the estrogen neoergosterol by direct peroxide cleavage Ray V. Lawrence and Walter H. Schuller pp 466 - 466; DOI: 10.1021/jm00287a033 |
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trans-2-Aminoethyl 2-acetoxycinnamates. Potential analgetic antiinflammatory agents Alex Gringauz pp 467 - 467; DOI: 10.1021/jm00287a034 |
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Derivatives of fluorene. 34. N1-acetyl-N2-fluorenylasparagines T. Lloyd Fletcher and Moses J. Namkung pp 467 - 467; DOI: 10.1021/jm00287a035 |
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The Androgens of the Testes R.E. Counsell pp 468 - 468; DOI: 10.1021/jm00287a900 |
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Structure and synthesis of the thyrotropin-releasing hormone K. Folkers, F. Enzmann, J. Boeler, C. Y. Bowers, and A. V. Schally pp 469 - 474; DOI: 10.1021/jm00288a001 |
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Synthesis of the thyrotropin-releasing hormone Karl Folkers, Jan Boeler, Jaw-Kang Chang, and Franz Enzmann pp 475 - 476; DOI: 10.1021/jm00288a002 |
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Synthetic thyrotropin-releasing hormone. Activity in men and women, specificity of action, inhibition by triiodothyronine, and activity orally K. Folkers, C. Y. Bowers, A. V. Schally, A. Kastin, A. Arimura, D. S. Schalch, C. Gual, and E. Castineda pp 477 - 481; DOI: 10.1021/jm00288a003 |
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Syntheses of pyroglutamylhistidylprolinamide and unusual mass fragmentation Karl Folkers, Jaw-Kang Chang, Hans Sievertsson, Conny Bogentoft, Bruce Currie, and G. Doyle Daves pp 481 - 483; DOI: 10.1021/jm00288a004 |
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Synthesis of analogs of the thyrotropin-releasing hormone and structure. Activity relations Karl Folkers, Jaw-Kang Chang, Hans Sievertsson, Bruce Currie, and Cyril Bowers pp 484 - 487; DOI: 10.1021/jm00288a005 |
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Linear polypeptides of a known primary structure. Synthesis and immunochemical studies of poly(L-glutamyl-L-tyrosyl-L-alanylglycyl)glycine-1-14C ethyl ester Brian John Johnson pp 488 - 489; DOI: 10.1021/jm00288a006 |
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Synthesis of [5-valine,7-N-methylalanine]-angiotensin II, a hypertensive peptide Harold A. Scheraga and Rudolf H. Andreatta pp 489 - 492; DOI: 10.1021/jm00288a007 |
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Lysophosphatidylethanolamine and 2-desoxylysophosphatidylethanolamine derivatives. 1. Potential renin inhibitors Francis R. Pfeiffer, Suzanne C. Hoke, Clara K. Miao, Ralph E. Tedeschi, Josephine Pasternak, Richard Hahn, Robert W. Erickson, Herman W. Levin, Charlotte A. Burton, and Jerry A. Weisbach pp 493 - 499; DOI: 10.1021/jm00288a008 |
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Potential folic acid antagonists. 4. Synthesis and dihydrofolate reductase inhibitory activities of 2,4,6-triamino-5-arylazopyrimidines D. J. Triggle, S. S. Chatterjee, D. R. Garrison, R. Kaprove, J. F. Moran, A. M. Triggle, and A. Wayne pp 499 - 501; DOI: 10.1021/jm00288a009 |
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Medium ring homologs of proline as potential amino acid antimetabolites H. T. Nagasawa, J. A. Elberling, P. S. Fraser, and N. S. Mizuno pp 501 - 508; DOI: 10.1021/jm00288a010 |
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Inhibition of sodium- and potassium-dependent adenosine triphosphatase by cardenolide alkylating agents Hanley N. Abramson and Jung-Sook K. Cho pp 509 - 511; DOI: 10.1021/jm00288a011 |
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.beta.-Adrenergic blocking agents. 10. (3-Amino-2-hydroxypropoxy)anilides Leslie Harold Smith, A. F. Crowther, and R. Howe pp 511 - 513; DOI: 10.1021/jm00288a012 |
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Physical and pharmacological properties of an irreversible local anesthetic Gerald M. Rosen, Seymour Ehrenpreis, Thomas W. Mittag, and James F. Stubbins pp 514 - 516; DOI: 10.1021/jm00288a013 |
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General anesthetics. 1. Halogenated methyl ethyl ethers as anesthetic agents Ross C. Terrell, Louise Speers, Alex J. Szur, John Treadwell, and Thomas R. Ucciardi pp 517 - 519; DOI: 10.1021/jm00288a014 |
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Anxiolytic sedatives. 1. Synthesis and pharmacology of benzo[6,7]-1,4-diazepino[5,4-b]oxazole derivatives and analogs Ryuji Tachikawa, Tetsuo Miyadera, Atsusuke Terada, Mitsunobu Fukunaga, Yoichi Kawano, Toshiharu Kamioka, Chihiro Tamura, and Hiromu Takagi pp 520 - 526; DOI: 10.1021/jm00288a015 |
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Synthesis and biological properties of certain trichloromethyl compounds Laszlo L. Darko pp 527 - 528; DOI: 10.1021/jm00288a016 |
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Synthesis and antimicrobial evaluation of some 5-(5-nitrofurylidene)rhodanines, 5-(5-nitrofurylidene)thiazolidine-2,4-diones, and their vinylogs S. K. Mallick, A. R. Martin, and R. G. Lingard pp 528 - 532; DOI: 10.1021/jm00288a017 |
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Antimalarials. "Distal" hydrazine derivatives of 7-chloroquinoline Tara Singh, John F. Hoops, John H. Biel, Wallace K. Hoya, Robert George Stein, and Deanna R. Cruz pp 532 - 535; DOI: 10.1021/jm00288a018 |
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Antiviral agents. 2. Structure-activity relations of compounds related to 1-adamantanamine Paul E. Aldrich, Edward C. Hermann, Walter E. Meier, Marvin Paulshock, William W. Prichard, Jack Austin Synder, and John C. Watts pp 535 - 543; DOI: 10.1021/jm00288a019 |
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8-Azatheophylline and its derivatives as coronary vasodilators D. S. Bariana pp 543 - 545; DOI: 10.1021/jm00288a020 |
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Synthesis of 1-amino-2-hydroxycyclopentanecarboxylic acid Charles G. Skinner and John D. Huddle pp 545 - 546; DOI: 10.1021/jm00288a021 |
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Antiviral agents. 1. Benzothiazole and benzoxazole analogs of 2-(.alpha.-hydroxybenzyl)benzimidazole W. A. Skinner, F. Gualtiere, G. Brody, and A. H. Fieldsteel pp 546 - 549; DOI: 10.1021/jm00288a022 |
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3- and 4-Carbazole dialkylaminocarbinols as potential antimalarial agents Joseph I. DeGraw, Vernon H. Brown, and Monsoor Keyanpour-Rad pp 549 - 550; DOI: 10.1021/jm00288a023 |
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Antimalarial agents. 7. Compounds related to 4,4'-bis(aminophenyl) sulfone Ivan C. Popoff, Gopal H. Singhal, and Allan R. Engle pp 550 - 551; DOI: 10.1021/jm00288a024 |
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Analgetic and anticonvulsant activity of some 2- and 4-pyridyl ketones J. Gearien, Eugene Frank, M. Megahy, and C. Pokorny pp 551 - 553; DOI: 10.1021/jm00288a025 |
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Central nervous system depressive activity of some amides of tryptamine Beng T. Ho, Rong An, Michael B. Noel, and L. Wayne Tansey pp 553 - 554; DOI: 10.1021/jm00288a026 |
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Quinuclidine analogs of tobacco alkaloids Alfred Burger and F. D. Reed pp 554 - 556; DOI: 10.1021/jm00288a027 |
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Deamino-D-oxytocin Vincent Du Vigneaud and George Flouret pp 556 - 557; DOI: 10.1021/jm00288a028 |
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.alpha.-Bromo- and .alpha.-chloropyridylalanines S. J. Norton and P. Timothy Sullivan pp 557 - 558; DOI: 10.1021/jm00288a029 |
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Quaternary ammonium salts of tertiary aminoalkyl amides Robert R. Mod, Frank C. Magne, Evald L. Skau, and Gene Sumrell pp 558 - 560; DOI: 10.1021/jm00288a030 |
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Stereochemical studies on medicinal agents. 10. Role of chirality in .alpha.-adrenergic receptor blockage by (+)- and (-)-phenoxy benzamine hydrochloride P. S. Portoghese, T. N. Riley, and J. W. Miller pp 561 - 564; DOI: 10.1021/jm00289a001 |
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Synthesis and analgetic activity of 3- and 4-methyl-6,7-benzomorphans Robert T. Parfitt and Susan M. Walters pp 565 - 568; DOI: 10.1021/jm00289a002 |
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Vitamin B6 analogs. 4. 4-Deoxyisopyridoxal and the phosphonic acid analog of 4-deoxypyridoxine phosphate Robert F. Struck, Y. Fulmer Shealy, and John A. Montgomery pp 568 - 571; DOI: 10.1021/jm00289a003 |
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Alkaloid studies. 7. Reactions of 18-hydroxymethyleneyohimban-17-one and the preparation of yohimbano[17,18-c and 18,17-d]pyrazoles Leon Goldman, J. Donald Albright, Natalie H. Conroy, and Arnold C. Osterberg pp 571 - 574; DOI: 10.1021/jm00289a004 |
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Novel pharmacological activity of a series of substituted pyridines Donald E. Butler, Paul Bass, Ivan C. Nordin, Frederick P. Hauck, and Yvon J. L'Italien pp 575 - 579; DOI: 10.1021/jm00289a005 |
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Synthesis and structure-activity relations of fibrinolytic bis(tetrahydroisoquinolines) Leonard J. Fliedner, Joseph M. Schor, Melvyn J. Myers, and Irwin J. Pachter pp 580 - 583; DOI: 10.1021/jm00289a006 |
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Synthesis of 1,2,3,4-tetrahydro-1,1,2,3,3,4,4-heptamethyl-6,7-dimethoxyisoquinoline and related compounds as potential hypotensive agents Jacob Finkelstein, Elliot Chiang, and Arnold Brossi pp 584 - 588; DOI: 10.1021/jm00289a007 |
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Central nervous system depressants. 9. Benzodiazepine sulfonamides Robert B. Moffett and Allan D. Rudzik pp 588 - 593; DOI: 10.1021/jm00289a008 |
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General anesthetics. 2. Halogenated methyl isopropyl ethers Louise Speers, Alex J. Szur, Ross C. Terrell, John Treadwell, and Thomas U. Ucciardi pp 593 - 595; DOI: 10.1021/jm00289a009 |
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Aromatic sulfonic acids as viral inhibitors. Structure-activity study using rhino, adeno 3, herpes simplex, and influenza viruses Stig Akerfeldt, Gertrud Westin, and Torsten Jansson pp 596 - 600; DOI: 10.1021/jm00289a010 |
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Synthesis of potential anticancer agents. 38. N-nitrosoureas. 4. Further synthesis and evaluation of haloethyl derivatives Thomas P. Johnston, George S. McCaler, Pamela S. Opliger, W. Russell Laster, and John A. Montgomery pp 600 - 614; DOI: 10.1021/jm00289a011 |
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Selectivity of action of alkylating agents and drug resistance. 4. Synthesis of tritium-labeled chlorambucil and a study of its cellular uptake by drug-sensitive and drug-resistant strains of the Yoshida ascites sarcoma in vitro Bridget T. Hill, Michael Jarman, and Kenneth R. Harrap pp 614 - 618; DOI: 10.1021/jm00289a012 |
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Bromomesaconic and bromocitraconic acids. Potential active site labeling reagents for dicarboxylic acid metabolizing enzymes Richard A. Laursen, Wei-Chiang Shen, and Kenneth G. Zahka pp 619 - 621; DOI: 10.1021/jm00289a013 |
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Nucleophilicity of some reactivators of phosphorylated acetylcholinesterase. 5 Sasson Cohen and Yacov Ashani pp 621 - 626; DOI: 10.1021/jm00289a014 |
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Comparative pharmacology of 5-hydroxytryptamine and its benzofuran, benzo[b]thiophen, and indene isosteres Roger M. Pinder, David M. Green, and Pamela B. J. Thompson pp 626 - 628; DOI: 10.1021/jm00289a015 |
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Synthesis and pharmacology of an epoxide derivative of ethacrynic acid Daniel A. Koechel, Ole Gisvold, and Edward J. Cafruny pp 628 - 629; DOI: 10.1021/jm00289a016 |
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Synthesis of some 3,7-dihydroxy-6-methyl-.DELTA.5-pregnene derivatives R. A. LeMahieu, A. Boris, M. Carson, and R. W. Kierstead pp 629 - 631; DOI: 10.1021/jm00289a017 |
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Angiotensin II analogs. 5. [2-Glycine]angiotensin II and related analogs Eugene C. Jorgensen, Graham C. Windridge, and Thomas Choy Lee pp 631 - 633; DOI: 10.1021/jm00289a018 |
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Antibacterial nitrofuran derivatives. 2. 5-Nitro-2-furaldehyde aminoacethydrazones E. Massarani, D. Nardi, A. Tajana, and L. Degen pp 633 - 635; DOI: 10.1021/jm00289a019 |
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Antibacterial nitrofuran derivatives. 3. 5-Nitro-2-furaldehyde piperazinoacylhydrazones E. Massarani, D. Nardi, S. Rossi, A. Tajana, and L. Degen pp 635 - 638; DOI: 10.1021/jm00289a020 |
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Synthetic antibacterials. 3. Nitrofurylvinyl-1,8-naphthyridine derivatives Fumio Yoneda, Sadao Nishigaki, Noriko Mizushima, and Hiroshi Takahashi pp 638 - 640; DOI: 10.1021/jm00289a021 |
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Linear polypeptides of a known primary structure. Synthesis and immunochemical studies of poly(O-methyl-L-tyrosyl-L-glutamyl-L-alanylglycyl)glycine-1-14C ethyl ester Brian J. Johnson and Francis Chen pp 640 - 641; DOI: 10.1021/jm00289a022 |
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Pyridoxine chemistry. 25. Analogs of vitamin B6 with reactive groups W. Korytnyk and B. Lachmann pp 641 - 643; DOI: 10.1021/jm00289a023 |
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Microsomal 3-hydroxylation of 1,4-benzodiazepines Neal Castagnoli, Wolfgang Sadee, and William Garland pp 643 - 645; DOI: 10.1021/jm00289a024 |
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Synthesis and pharmacology of some N-substituted derivatives of 1-amino-4,6-dimethylbenzocyclobutene Arthur A. Siciliano and Karl A. Nieforth pp 645 - 646; DOI: 10.1021/jm00289a025 |
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5-Benzoyl-1-methylpyrrole-2-acetic acids as antiinflammatory agents John R. Carson, Doris N. McKinstry, and Stewart Wong pp 646 - 647; DOI: 10.1021/jm00289a026 |
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Phosphorus-nitrogen compounds. 12. Phosphamidase studies. 2. N-alkylphosphoramidic acids Lindley A. Cates pp 647 - 649; DOI: 10.1021/jm00289a027 |
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Potential antidiabetics. 9. Biological activity of some pyrazoles H. G. Garg and Chandra Prakash pp 649 - 650; DOI: 10.1021/jm00289a028 |
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2,5-Dimethoxy-4-methylphenylalanine Roger M. Pinder and Keith Brewster pp 650 - 651; DOI: 10.1021/jm00289a029 |
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Progress in Drug Research Alfred Burger pp 652 - 652; DOI: 10.1021/jm00289a900 |
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Nucleoside Antibiotics Alfred Burger pp 652 - 652; DOI: 10.1021/jm00289a901 |
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Structure-activity relations in antifungal agents. A survey Corwin Hansch and Eric J. Lien pp 653 - 670; DOI: 10.1021/jm00290a001 |
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Crystal structure of dl-brompheniramine maleate {1-(p-bromophenyl)-1- (2-pyridyl)-3-N,N-dimethylaminopropane maleate} M. N. G. James and G. J. B. Williams pp 670 - 675; DOI: 10.1021/jm00290a002 |
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Steroidal androgen biosynthesis inhibitors G. E. Arth, A. A. Patchett, T. Jefopoulus, R. L. Bugianesi, L. H. Peterson, E. A. Ham, F. A. Kuehl, and N. G. Brink pp 675 - 679; DOI: 10.1021/jm00290a003 |
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Interdependence between physical parameters and selection of substituent groups for correlation studies Paul N. Craig pp 680 - 684; DOI: 10.1021/jm00290a004 |
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Inhibitors and stimulators of cholesterolgenesis enzymes. Structure-activity study in vitro of amino and selected nitrogen-containing analogs of 5.alpha.-cholestane-3.beta.,5.alpha.,6.beta.-triol Donald T. Witiak, Roger A. Parker, Mary E. Dempsey, and Mary C. Ritter pp 684 - 693; DOI: 10.1021/jm00290a005 |
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Potential folic acid antagonists. 5. Synthesis and biologic evaluation of N10-deazapteroic acid and N10-deazafolic acid and their 9,10-dehydro derivatives Robert F. Struck, Y. Fulmer Shealy, and John A. Montgomery pp 693 - 698; DOI: 10.1021/jm00290a006 |
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Muscarinic receptors. Derivatives of 7-oxabicyclo[2.2.1]heptane Wendel L. Nelson, David R. Allen, and Frank F. Vincenzi pp 698 - 702; DOI: 10.1021/jm00290a007 |
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Conformational study of catechol amine receptor sites. 7. Syntheses of erythro-and threo-3-amino-2-(3,4-dihydroxyphenyl)-2-butanol hydrochlorides and erythro- and threo-2-amino-3-(3,4-dihydroxyphenyl)butanehydrochlorides Edward E. Smissman and Ronald T. Borchardt pp 702 - 707; DOI: 10.1021/jm00290a008 |
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Acenaphthene chemistry. 2. Synthesis and antiinflammatory activity of 1-[2-(dimethylamino)ethyl]-2,2-dimethyl-1-acenaphthenecarboxamide Syemour D. Levine pp 707 - 709; DOI: 10.1021/jm00290a009 |
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Carbanilic acid esters of cyclic amino alcohols. 4. Esters of pyrrolidinols and piperidinols as local anesthetics Richard Dahlbom, J. Lars G. Nilsson, and Hans Sievertsson pp 710 - 714; DOI: 10.1021/jm00290a010 |
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2-(Alkenylamino)benzamides and related 1-(alkenyl)-4(1H)-quinazolinones as analgetics and antiinflammatories Michel Vincent, Jean C. Poignant, and Georges Remond pp 714 - 717; DOI: 10.1021/jm00290a011 |
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Conformational studies of amphetamine and medicinally important derivatives by nuclear magnetic resonance spectroscopy George A. Neville, Roxanne Deslauriers, Barry J. Blackburn, and Ian C. P. Smith pp 717 - 721; DOI: 10.1021/jm00290a012 |
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New series of semisynthetic rifamycins. N-substituted derivatives of 4-amino-4-deoxyrifamycin SV Renato Cricchio and Giovanni Tamborini pp 721 - 723; DOI: 10.1021/jm00290a013 |
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Prediction of the in vitro activity of sulfonamides synthesized from simple amines by use of electronic data obtained from the simple amines Joachim K. Seydel pp 724 - 729; DOI: 10.1021/jm00290a014 |
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Synthesis of compounds structurally related to poison ivy urushiol. 3. 3-n-Pentadecylcatechol and 3-n-alkylcatechols of varying side-chain length Charles R. Dawson and A. Peter Kurtz pp 729 - 732; DOI: 10.1021/jm00290a015 |
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Synthesis of compounds structurally related to poison ivy urushiol. 4. 3-(1-Alkyl)alkylcatechols of varying side-chain shape and flexibility Charles R. Dawson and A. Peter Kurtz pp 733 - 737; DOI: 10.1021/jm00290a016 |
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Synthesis and antihypertensive properties of some N-(guanidinoalkyl)pyrrolidines David Miller, Brian P. Curwain, Charles S. Fake, John L. Gordon, Minoo D. Mehta, Robert H. Poyster, and Eric A. Watts pp 737 - 742; DOI: 10.1021/jm00290a017 |
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Thiazolothiazoles. 3. Synthesis and biological evaluation of functionalized dialkyl derivatives from .gamma.,.gamma.,.gamma.',.gamma.'-tetramethylthiazolo[5,4-d]thiazole-2,5-dibutyronitrile Roger Ketcham and Sonia Mah pp 743 - 747; DOI: 10.1021/jm00290a018 |
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Synthesis of naturally occurring 6-ureidopurines and their nucleosides Girish B. Chheda and Chung Il Hong pp 748 - 753; DOI: 10.1021/jm00290a019 |
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Inhibitory action of .alpha.-(4-chlorophenoxy)-.alpha.-methylpropionic acid analogs on cholesterol biosynthesis and lipolysis in vitro Donald T. Witiak, Dennis R. Feller, Eugene S. Stratford, Robert E. Hackney, Ralph Nazareth, and Gwen Wagner pp 754 - 757; DOI: 10.1021/jm00290a020 |
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6-Chlorochroman-2-carboxylic acids. Synthesis and biological evaluation as antagonists for cholesterol biosynthesis and lipolysis in vitro Donald T. Witiak, Eugene S. Stratford, Ralph Nazareth, Gwen Wagner, and Dennis R. Feller pp 758 - 766; DOI: 10.1021/jm00290a021 |
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Griseofulvin analogs. 9. Griseofulvin analogs derived from transformations of 5'-formylgriseofulvin Howard Newman, Thomas L. Fields, and Robert B. Angier pp 767 - 769; DOI: 10.1021/jm00290a022 |
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Synthesis and biological response of some 3-iminoprogestins Arvin P. Shroff, R. P. Blyte, and J. L. McGuire pp 769 - 770; DOI: 10.1021/jm00290a023 |
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.beta.-Lactam antimicrobial agents which possess antifungal activity Lee C. Cheney, William J. Gottstein, Ann H. Eachus, Peter F. Misco, Martin Misiek, and Kenneth E. Price pp 770 - 772; DOI: 10.1021/jm00290a024 |
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Insect chemosterilants. 10. Substituted dithiobiurets A. B. Borkovec, J. E. Oliver, S. C. Chang, and R. T. Brown pp 772 - 773; DOI: 10.1021/jm00290a025 |
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Vitamin B6 analogs. Improved synthesis of 3-hydroxypyridine-4-carboxaldehyde Marion H. O'Leary and James R. Payne pp 773 - 774; DOI: 10.1021/jm00290a026 |
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Peptides with terminal tyrosyl and phenylalanyl groups Joseph A. Skorcz pp 775 - 776; DOI: 10.1021/jm00290a027 |
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Analogs of bradykinin containing .beta.-2-thienyl-L-alanine John Morrow Stewart and Floyd W. Dunn pp 779 - 781; DOI: 10.1021/jm00291a001 |
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Inhibitors of platelet aggregation. 2. 9-{[(Dialkylamino)alkyl]thio}-3-(dimethylamino)acridines and related acridine derivatives Edward F. Elslager, Neil F. Haley, J. R. McLean, S. C. Perricone, Doris Potoczak, H. Veloso, Donald F. Worth, and R. H. Wheelock pp 782 - 788; DOI: 10.1021/jm00291a002 |
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Aromatic amino acid hydroxylase inhibitors. 2. 3-Alkyl-.alpha.-methyltyrosines R. E. Counsell, P. Desai, A. Ide, P. G. Kulkarni, P. A Weinhold, and V. B. Rethy pp 789 - 792; DOI: 10.1021/jm00291a003 |
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Irreversible enzyme inhibitors. 183. Proteolytic enzymes. 18. Inhibitors of guinea pig complement derived by quaternization of phenylalkylpyridines with .alpha.-bromomethylbenzenesulfonyl fluorides B. R. Baker and Michael H. Doll pp 793 - 799; DOI: 10.1021/jm00291a004 |
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Irreversible enzyme inhibitors. 184. Affinity column for purification of rat liver guanine deaminase and xanthine oxidase B. R. Baker and Hans U. Siebeneick pp 799 - 801; DOI: 10.1021/jm00291a005 |
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Irreversible enzyme inhibitors. 185. Active-site-directed irreversible inhibitors of guanine deaminase derived from 9-phenylguanine bearing a terminal sulfonyl fluoride. 2 B. R. Baker and Hans U. Siebeneick pp 802 - 805; DOI: 10.1021/jm00291a006 |
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Irreversible enzyme inhibitors. 186. Irreversible inhibitors of the C'la component of complement derived from m-(phenoxypropoxy)benzamidine by bridging to a terminal sulfonyl fluoride B. R. Baker and Michael Cory pp 805 - 808; DOI: 10.1021/jm00291a007 |
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Irreversible enzyme inhibitors. 187. Bulk tolerance with inhibitors of guanosine phosphorylase B. R. Baker and James C. Schaeffer pp 809 - 812; DOI: 10.1021/jm00291a008 |
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Irreversible enzyme inhibitors. 188. Inhibition of mammalian thymidine phosphorylase B. R. Baker and James L. Kelley pp 812 - 816; DOI: 10.1021/jm00291a009 |
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Substituted hydroxylaminopurines and related derivatives. Synthesis and screening tests Alfredo Giner-Sorolla and Joseph H. Burchenal pp 816 - 819; DOI: 10.1021/jm00291a010 |
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Xylo- and arabinofuranosylthioguanine and related nucleosides derived from 2-acetamido-6-chloropurine William W. Lee, Abelardo P. Martinez, Robert W. Blackford, Victor J. Bartuska, Elmer J. Reist, and Leon Goodman pp 819 - 823; DOI: 10.1021/jm00291a011 |
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Calculation of the .pi.-electron "ring current" properties of some carcinogenic, heptacyclic, condensed, benzenoid hydrocarbons Roger B. Mallion pp 824 - 826; DOI: 10.1021/jm00291a012 |
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Steroids and steroidases. 10. Potentially antitumor active androstane compounds containing C-17 nitrogen mustard functions J. Bryan Jones, David J. Adam, and Jeffrey D. Leman pp 827 - 833; DOI: 10.1021/jm00291a013 |
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Stereochemical aspects of antihistamine action. 4. Absolute configuration of carbinoxamine antipodes G. Hite, V. Barouh, H. Dall, and D. Patel pp 834 - 836; DOI: 10.1021/jm00291a014 |
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Aryloxyalkylamines, N-arylethylenediamines, and related compounds as anorectic agents C. J. Sharpe, R. S. Shadbolt, G. R. Brown, A. Ashford, and J. W. Ross pp 836 - 842; DOI: 10.1021/jm00291a015 |
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Microbiological and chemical modification of N-benzoyl-N,2,3,3-tetramethyl-exo-2-norbornanamine (N-benzoylmecamylamine) Milton E. Herr, Herbert C. Murray, and Gunther S. Fonken pp 842 - 845; DOI: 10.1021/jm00291a016 |
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Central nervous system activities of thiolactams and lactams. Structure-activity correlations E. J. Lien, L. L. Lien, and G. L. Tong pp 846 - 848; DOI: 10.1021/jm00291a017 |
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Benzazepinones. Synthesis of the monoaza analog of diazepam, and the correct structure of the benzoylpropionanilide cyclization product Bernard Loev, Richard B. Greenwald, Marjorie M. Goodman, and Charles L. Zirkle pp 849 - 852; DOI: 10.1021/jm00291a018 |
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Synthesis of acyloxyalkylbarbiturates as potential long-acting central nervous system depressants Edward E. Smissman, Robert A. Robinson, and Marcia A. Buckwalter pp 853 - 855; DOI: 10.1021/jm00291a019 |
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Isoxazole chemistry. 5. N-Alkylation and N-acylation of 5-amino-3-(5-nitro-2-furyl)isoxazoles R. G. Micetich, R. Raap, and C. G. Chin pp 856 - 860; DOI: 10.1021/jm00291a020 |
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Synthesis of indoles from 4-oxo-4,5,6,7-tetrahydroindoles. 4. Tricyclic heterocycles William A. Remers, Reta H. Roth, and Martin J. Weiss pp 860 - 862; DOI: 10.1021/jm00291a021 |
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Antimalarial activity of guanylhydrazone salts of aromatic ketones. 2. Development of active polyhalo derivatives Frederic A. French, Jefferson R. DoAmaral, Erwin J. Blanz, and Douglas A. French pp 862 - 866; DOI: 10.1021/jm00291a022 |
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2,4-Diamino-6-arylethylpteridines as Streptococcus faecium growth inhibitors Joseph I. DeGraw, Vernon H. Brown, Roy L. Kisliuk, and Yvette Gaumont pp 866 - 867; DOI: 10.1021/jm00291a023 |
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Biologically oriented organic sulfur chemistry. 8. Structure-activity relations of penicillamine analogs and derivatives L. Field, B. J. Sweetman, M. M. Vestling, S. T. Ticaric, P. L. Kelly, P. Merryman, and I. A. Jaffe pp 868 - 872; DOI: 10.1021/jm00291a024 |
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Receptor site labeling through functional groups. Barbital and amphetamine derivatives Edward M. Kosower, Tetsuo Miyadera, and Nechama S. Kosower pp 873 - 878; DOI: 10.1021/jm00291a025 |
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Tetracyclic quinazolinone derivatives Goetz E. Hardtmann, Bruno S. Heugi, John H. Gogerty, Louis C. Iorio, and H. William Barnes pp 878 - 882; DOI: 10.1021/jm00291a026 |
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Nucleic acids. 12. Synthesis of the L enantiomer of 1-.beta.-arabinofuranosylcytosine and of O2, O2'-anhydro-1-.beta.-D-arabinofuranosylcytosine William J. Wechter, Duane T. Gish, and Gary L. Neil pp 882 - 883; DOI: 10.1021/jm00291a027 |
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4(5)-(2-Amino-1-hydroxyalkyl)imidazoles Alfred Burger and Manuelo Bernabe pp 883 - 885; DOI: 10.1021/jm00291a028 |
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Potential inhibitors of protein biosynthesis G. Hite, A. P. Grollman, and S. Rosen pp 885 - 887; DOI: 10.1021/jm00291a029 |
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Potential anticancer agents. Nitrogen mustards of aminophenylthiazoles C. V. Deliwala, J. D. Modi, and S. S. Sabnis pp 887 - 888; DOI: 10.1021/jm00291a030 |
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Synthesis and pharmacology of some dimethoxy-substituted indanamines as potential hypoglycemic agents. 1-Methyl-2-[(dialkylamino)methyl]-5,6-dimethoxyindans Samir C. Lahiri and Balai Pathak pp 888 - 889; DOI: 10.1021/jm00291a031 |
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Synthesis of some 1-piperazinecarboxalic acid ethyl ester derivatives as possible antifilarial and antihypertensive agents Prabhash C. Das, B. B. Patra, S. B. Chaudhuri, U. P. Basu, B. N. Kolay, and S R. Maitra pp 890 - 891; DOI: 10.1021/jm00291a032 |
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Optical isomers of mepivacaine and bupivacaine Benjamin F. Tullar pp 891 - 892; DOI: 10.1021/jm00291a033 |
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2-Aminoindan-2-carboxylic acids. Potential tyrosine hydroxylase inhibitors Rober M. Pinder, Brian H. Butcher, David A. Buxton, and David J. Howells pp 892 - 893; DOI: 10.1021/jm00291a034 |
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Synthesis and peripheral vasodilator activity of .alpha.-[1-(4-piperidylamino)alkyl]benzyl alcohols John L. Hughes, Jay K. Seyler, Carroll M. Smith, and Pedro D. Luna pp 894 - 895; DOI: 10.1021/jm00291a035 |
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Absolute configuration of the optical isomers of salbutamol D. Hartley and D. Middlemiss pp 895 - 896; DOI: 10.1021/jm00291a036 |
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Synthesis and local anesthetic activity of N-diethylaminoacetyl derivatives of naphthylalkylamines Gianfranco Pala, Arturo Donetti, Antonio Mantegani, and Camillo Bianchi pp 896 - 897; DOI: 10.1021/jm00291a037 |
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5-Cyclohexylmethyl-5-arylhydantoins Jorge R. Barrio, Maria Del Carmen G. Barrio, and Marcelo J. Vernengo pp 898 - 898; DOI: 10.1021/jm00291a038 |
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Influence of Hydrophobic Character on the Relative Rate of Oxidation of Drugs by Rat Liver Microsomes Yvonne C. Martin pp 777 - 779; DOI: 10.1021/jm00291a600 |
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Angiotensin II analogs. 6. Stereochemical factors in the 5 position influencing pressor activity. 1 Eugene C. Jorgensen, Sambasiva R. Rapaka, Graham C. Windridge, and Thomas C. Lee pp 899 - 903; DOI: 10.1021/jm00292a001 |
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Angiotensin II analogs. 7. Stereochemical factors in the 5 position influencing pressor activity. 2 Eugene C. Jorgensen, Sambasiva R. Rapaka, Graham C. Windridge, and Thomas C. Lee pp 904 - 906; DOI: 10.1021/jm00292a002 |
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Synthesis and antihypertensive activity of 2-arylamino-1-azacycloalkenes Fred M. Hershenson and Leonard F. Rozek pp 907 - 909; DOI: 10.1021/jm00292a003 |
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Antihypertensive and monoamine oxidase inhibitory activity of some azacycloaklyl-substituted benzaldehyde hydrazone derivatives T. George, C. L. Kaul, R. S. Grewal, and D. V. Mehta pp 909 - 913; DOI: 10.1021/jm00292a004 |
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Antihypertensive and monoamine oxidase inhibitory activity of some derivatives of 3-formyl-4-oxo-4H-pyrido[1,2-a]pyrimidine T. George, C. L. Kaul, R. S. Grewal, and R. Tahilramani pp 913 - 915; DOI: 10.1021/jm00292a005 |
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Novel schistosomicides. S-2-{[2-(2-Thiazolylcarbamoyl)ethyl]amino}ethyl hydrogen thiosulfate and related compounds Roger D. Westland, Leslie M. Werbel, John R. Dice, Joyce L. Holmes, and Barbara G. Zahm pp 916 - 920; DOI: 10.1021/jm00292a006 |
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Antimalarial phenathrene amino alcohols. 1. Fluorine-containing 3- and 6-substituted 9-phenanthrenemethanols Edward A. Nodiff, Keiichi Tanabe, Christoph Seyfried, Shin Matsuura, Yasuaki Kondo, Eugene H. Chen, and Mahesh P. Tyagi pp 921 - 925; DOI: 10.1021/jm00292a007 |
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Antimalarials. 7. Bis(trifluoromethyl)-.alpha.-(2-piperidyl)-4-quinolinemethanols R. E. Lutz, C. J. Ohnmacht, and A. R. Patel pp 926 - 928; DOI: 10.1021/jm00292a008 |
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Potential filaricides. 5. 3-Ethyl-8-methyl-1,3,8-triazabicyclo[4.4.0]decan-2-one, a new antifilarial agent Nitya Anand, Ranjna Saxena, Satyavan Sharma, and R. N. Iyer pp 929 - 931; DOI: 10.1021/jm00292a009 |
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Deuterium isotope effect in chloramphenicol action Eberhard Kutter and Hans Machleidt pp 931 - 934; DOI: 10.1021/jm00292a010 |
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Chemotherapeutic nitro heterocycles. 7. Substituted 5-alkylthiomethyl-3-(5-nitro-2-imidazolyl)methyleneamino-2-oxazolidinones C. Rufer, H. J. Kessler, and E. Schroeder pp 934 - 935; DOI: 10.1021/jm00292a011 |
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Mitosis-inhibiting natural products. 24. Synthesis and antimitotic activity of glycosidic lignan derivatives related to podophyllotoxin C. Keller-Juslen, M. Kuhn, A. Von Wartburg, and H. Staehelin pp 936 - 940; DOI: 10.1021/jm00292a012 |
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Carcinogenic and adrenocorticolytic derivatives of benz[a]anthracene John Pataki, Carol Duguid, Peter W. Rabideau, Howard Huisman, and Ronald G. Harvey pp 940 - 945; DOI: 10.1021/jm00292a013 |
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Specificity in enzyme inhibition. 1. Synthesis of 4-(4-imidazolyl)-3-amino-2-butanone, 4-(4-imidazolyl)-3-acetamido-2-butanone, and 4-(4-imidazolylmethyl 2,5-dimethyloxazole for assay as inhibitors of histidine decarboxylase Edward E. Smissman and James A. Weis pp 945 - 947; DOI: 10.1021/jm00292a014 |
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Pyridoxine chemistry. 26. 5-Homopyridoxals, 5-thiopyridoxal, and related compounds. Synthesis, tautomerism, and biological properties W. Korytnyk and H. Ahrens pp 947 - 952; DOI: 10.1021/jm00292a015 |
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Antiestrogenic and antifertility compounds. 4. 1,1,2-Triarylalkan-1-ols and 1,1,2-triarylalk-1-enes containing basic ether groups D. J. Collins, J. J. Hobbs, and C. W. Emmens pp 952 - 957; DOI: 10.1021/jm00292a016 |
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Heterocyclic steroids. 2. Synthesis and androgenic activity of A-ring oxaandrostanes Manfred E. Wolff and Galal Zanati pp 958 - 961; DOI: 10.1021/jm00292a017 |
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Heterocyclic steroids. 3. Androgen having three heteroatoms in ring A Manfred E. Wolff and Galal Zanati pp 961 - 962; DOI: 10.1021/jm00292a018 |
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Antiulcer agents. p-Aminobenzamido aromatic compounds Robert B. Moffett, Andre Rober, and Louis L. Skaletzky pp 963 - 968; DOI: 10.1021/jm00292a019 |
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Metabolism of 3-(.alpha.,.alpha.,.alpha.-trifluoro-m-tolyloxy)-1,2-propanediol 1-carbamate in man Arlington A. Forist, Donald R. Buhler, Harry Harpootlian, and Ray W. Judy pp 969 - 971; DOI: 10.1021/jm00292a020 |
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Synthesis and analgesic properties of compounds containing an exocyclic basic center J. V. Greenhill pp 971 - 973; DOI: 10.1021/jm00292a021 |
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Antiinflammatory 3,4-dihydro-2-alkyl-3-oxo-2H-1,2-benzothiazine-4-carboxamide 1,1-dioxides Joseph G. Lombardino and Edward H. Wiseman pp 973 - 977; DOI: 10.1021/jm00292a022 |
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Phenacylthioimidazolines and 3-aryl-5,6-dihydroimidazo[2,1-b]thiazoles with antidepressant activity C. J. Sharpe, R. S. Shadbolt, A. Ashford, and J. W. Ross pp 977 - 982; DOI: 10.1021/jm00292a023 |
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Chemistry and pharmacology of 5-methylene-4-substituted dibenzo[.alpha.,d]cycloheptenes Leslie G. Humer, Ferenc Herr, and Marie P. Charest pp 982 - 985; DOI: 10.1021/jm00292a024 |
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cis-1-[2-(p-Anisidinomethyl)cyclohexyl]piperidine and related compounds. Oral hypoglycemic agents Ronald H. Rynbrandt, Fredericka L. Schmidt, and Jacob Szmuszkovicz pp 985 - 987; DOI: 10.1021/jm00292a025 |
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Heterocyclic systems. 1. 1-Substituted 1,2-dihydro-2-nitroiminopyridines John P. Paolini and Louis J. Lendvay pp 988 - 990; DOI: 10.1021/jm00292a026 |
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Antibacterial nitrofuran derivatives. 4. 5-Nitro-2-furaldehyde hydrazoniumacethydrazones E. Massarani, D. Nardi, R. Pozzi, and L. Degen pp 990 - 992; DOI: 10.1021/jm00292a027 |
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New antibacterial quinoxaline N,N-dioxide derivatives Gerald Berkelhammer and Peter H. Gund pp 992 - 992; DOI: 10.1021/jm00292a028 |
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Synthetic biologically active polymers. 9. Comparison of antimalarial activity in copolymers containing common sulfonamide monomers but different comonomers L. Guy Donaruma, John R. Dombroski, and John Razzano pp 993 - 993; DOI: 10.1021/jm00292a029 |
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Antihistomonal activity of ipronidazole and closely related nitroimidazoles A. Brossi, M. Hoffer, M. Mitrovic, and A. Beaman pp 993 - 994; DOI: 10.1021/jm00292a030 |
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Biologically oriented organic sulfur chemistry. 9. Carbonyl and thiocarbamoyl disulfides as inhibitory agents for Histoplasma capsulatum Lamar Field, Wayne S. Hanley, and Ilda McVeigh pp 995 - 996; DOI: 10.1021/jm00292a031 |
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Syntheses and screening of some trifluoromethyl pyrazoles Henry V. Secor and J. Fred. DeBardeleben pp 997 - 998; DOI: 10.1021/jm00292a032 |
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Structure of the diuretic merbaphen E. M. Schultz, J. B. Bicking, S. J. DeSolms, and G. E. Stokker pp 998 - 999; DOI: 10.1021/jm00292a033 |
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Metal chelate steroid analogs. 2. [7-Amino-8-(aminomethyl)-1,2,3,4,4a,4b,5,6,7,8,8a,9-dodecahydro-4a,7-dimethyl-2-phenanthrol] bis(ethylenediamine)cobalt(3+) trichloride .beta.-acetate (ester) L. Guy Donaruma and Patricia U. Flath pp 999 - 1000; DOI: 10.1021/jm00292a034 |
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Synthesis and hypoglycemic activity of 3-aryl(or pyridyl)-5-alkyl(or aryl)amino-1,3,4-thiadiazoles and some sulfonylurea derivatives of 4H-1,2,4-triazoles C. V. Deliwala, M. Y. Mhasalkar, M. H. Shah, P. D. Pilankar, S. T. Nikam, and K. G. Anantanarayanan pp 1000 - 1003; DOI: 10.1021/jm00292a035 |
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Potential acetylcholinesterase reactivators. p.p'-Biphenyl and 1,4-benzene disubstituted oximes C. F. Barfknect, F. W. Benz, and J. P. Long pp 1003 - 1004; DOI: 10.1021/jm00292a036 |
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Synthesis and pharmacological activity of dialkylaminoethyl esters and amides of phenylmercaptoacetic acid and its derivatives G. Tsatsas, E. Costakis, W. Benson, and S. A. Ferguson pp 1004 - 1005; DOI: 10.1021/jm00292a037 |
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Neuropharmacological profile of 1-azaphenothiazine-10-thiolcarboxylates Edward R. Atkinson, Pamela L. Russ, Margaret A. Tucker, and Franklin J. Rosenberg pp 1005 - 1007; DOI: 10.1021/jm00292a038 |
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Central nervous system active butyrophenones. 1. Unsaturated analogs of .gamma.-aminobutyrophenones Samuel J. Dominianni, Richard P. Pioch, and Ronald L. Young pp 1008 - 1009; DOI: 10.1021/jm00292a039 |
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Central nervous system active butyrophenones. 2. Methyl-branched .gamma.-aminobutyrophenones Samuel J. Dominianni, Richard P. Pioch, Ronald L. Young, and Patrick J. Stimart pp 1009 - 1011; DOI: 10.1021/jm00292a040 |
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Synthesis and analgesic activity of 1,5-methano-3-methyl-1,2,3,4,5,6-hexahydro-3-benzazocines Lewis A. Walter, Wei K. Chang, and Robert I. Taber pp 1011 - 1013; DOI: 10.1021/jm00292a041 |
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Synthesis and pharmcological effects of some alkyl-, aryl, and aralkylsydnonimines V. Z. Gorkin, V. G. Yashunskii, M. D. Mashkovskii, R. A. Al'tshuler, I. V. Verevkina, and L. E. Kholodov pp 1013 - 1015; DOI: 10.1021/jm00292a042 |
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Quaternary isothiazolylpyridinium salts. Oral hypoglycemic agents Gretchen E. Wiegand, Victor J. Bauer, S. R. Safir, D. A. Blickens, and S. J. Riggi pp 1015 - 1016; DOI: 10.1021/jm00292a043 |
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Synthesis of new urethans. p-Cyclohexylsulfamoyl and p-piperidinosulfonylcarbanilic acid esters I. Lalezari and H. Golgolab pp 1017 - 1017; DOI: 10.1021/jm00292a044 |
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Aldehyde disubstituted aminoacethydrazones as potential hypertensive agents A. Tajana and R. Pozzi pp 1017 - 1020; DOI: 10.1021/jm00292a045 |
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1-Substituted 3,3-dimethylspiro[indoline-2,3-thietane] 1',1'-dioxides derived from 2-methyleneindolines Charles H. Tilford pp 1020 - 1021; DOI: 10.1021/jm00292a046 |
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Evaluation of carbazoles as antifungal agents Boris Weinstein and K. C. Das pp 1021 - 1021; DOI: 10.1021/jm00292a047 |
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Synthesis of L-dope (3,4-dihydroxyphenyl-L-alanine) Hiromasa Nakamoto, Masakazu Aburatani, and Mitsuru Inagaki pp 1021 - 1021; DOI: 10.1021/jm00292a048 |
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Phosphorus-nitrogen compounds. 13. Methoxyethyl and propylamine derivatives L. A. Cates and E. K. Ryu pp 1022 - 1022; DOI: 10.1021/jm00292a049 |
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Thyroxine analogs. 20. Substituted 1- and 2-naphthyl ethers of 3,5-diiodotyrosine Eugene C. Jorgensen and Peter Slade pp 1023 - 1026; DOI: 10.1021/jm00293a001 |
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Coenzyme Q. 114. Biosynthesis of coenzymes Q by malarial parasites. 2. Coenzyme Q synthesis in blood cultures of monkeys infected with malarial parasites (Plasmodium falciparum and P. knowlesi) Jerome V. Schnell, Wasim A. Siddiqui, Quentin M. Geiman, Frederick S. Skelton, Kenneth D. Lunan, and Karl Folkers pp 1026 - 1029; DOI: 10.1021/jm00293a002 |
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Coenzyme Q. 136. Synthesis of new 5,8-quinolinequinones as inhibitors of coenzyme Q and as antimalarials Thomas H. Porter, Frederick S. Skelton, and Karl Folkers pp 1029 - 1033; DOI: 10.1021/jm00293a003 |
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Schistosomicides. 1. Derivatives of 2-aminomethyl-1,2,3,4-tetrahydroquinoline C. A. R. Baxter and H. C. Richards pp 1033 - 1042; DOI: 10.1021/jm00293a004 |
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Synthesis of aminoethyl derivatives of .alpha.,.omega.-alkylenediamines and structure-activity relations for the polyamine-bovine plasma amine oxidase system Mervyn Israel and Edward J. Modest pp 1042 - 1047; DOI: 10.1021/jm00293a005 |
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6-Amino derivatives of stigmastanol and cholestanol H. Pinhas, A. Loiseau, A. Krikorian-Manoukian, D. Courmarcel, N. P. Buu-Hoi, and P. Jacquignon pp 1048 - 1049; DOI: 10.1021/jm00293a006 |
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[2,4-Dileucine]oxytocin. Polypeptide with natriuretic and diuretic activities, and an inhibitor of the oxytocic response of oxytocin Victor J. Hruby and W. Y. Chan pp 1050 - 1051; DOI: 10.1021/jm00293a007 |
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Synthesis of 1-methyl-1-(substituted benzyl)hydrazines Donald E. Butler, Susan M. Alexander, John W. McLean, and Linda B. Strand pp 1052 - 1054; DOI: 10.1021/jm00293a008 |
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Synthesis and hypotensive activity of benzamidopiperidylethylindoles J. L. Archibald, B. J. Alps, J. F. Cavalla, and J. L. Jackson pp 1054 - 1059; DOI: 10.1021/jm00293a009 |
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Synthesis and hypotensive properties of new 4-aminoquinolines George C. Wright, Edward J. Watson, Frank F. Ebetino, Guy Lougheed, Benjamin F. Stevenson, Alexander Winterstein, Robert K. Bickerton, Robert P. Halliday, and Donald T. Pals pp 1060 - 1066; DOI: 10.1021/jm00293a010 |
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Quaternary pilocarpine derivatives acting as acetylcholine antagonists A. Ben Bassat, D. Lavie, H. Edery, and G. Porath pp 1066 - 1069; DOI: 10.1021/jm00293a011 |
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Benzimidazo[2,1-b]quinazolin-12-ones. New class of potent immunosuppressive compounds W. H. W. Lunn, R. W. Harper, and R. L. Stone pp 1069 - 1071; DOI: 10.1021/jm00293a012 |
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Synthesis and antiinflammatory activity of tert-aminomethylbenzophenones Robert Coombs, William J. Houlihan, Jeffery Nadelson, and Edward I. Takesue pp 1072 - 1074; DOI: 10.1021/jm00293a013 |
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Derivatives of 2-aminooxazoles showing antiinflammatory activity George Crank and Michael J. Foulis pp 1075 - 1077; DOI: 10.1021/jm00293a014 |
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6-Phenyl-4H-s-triazolo[4,3-a][1,4]benzodiazepines which have central nervous system depressant activity Jackson B. Hester, Allan D. Rudzik, and Bharat V. Kamdar pp 1078 - 1081; DOI: 10.1021/jm00293a015 |
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Molecular orbital calculations on coumarins and the induction of drug-metabolizing enzymes R. W. Wald and G. Feuer pp 1081 - 1084; DOI: 10.1021/jm00293a016 |
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Interaction of ergothioneine with metal ions and metalloenzymes David P. Hanlon pp 1084 - 1087; DOI: 10.1021/jm00293a017 |
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Central nervous system agents. 1. Synthesis of diphenyl-tert-aminopropanols Robert B. Moffett, Richard E. Strube, and Louis Skaletzky pp 1088 - 1100; DOI: 10.1021/jm00293a018 |
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Central nervous system agents. 2. Synthesis of diphenyl primary and secondary aminopropanols Robert B. Moffett and Timothy L. Pickering pp 1100 - 1106; DOI: 10.1021/jm00293a019 |
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Central nervous system agents. 3. Structure-activity relation of a series of diphenylaminopropanols Huch H. Keasling and Robert B. Moffett pp 1106 - 1111; DOI: 10.1021/jm00293a020 |
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Synthesis of 1-.beta.-L-arabinofuranosylcytosine, the enantiomer of cytosine arabinoside Richard L. Tolman and Roland K. Robins pp 1112 - 1112; DOI: 10.1021/jm00293a021 |
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Antitumor activity of some phosphatidyl nitrogen mustard derivatives Joseph G. Turcotte and Gajanan P. Hedge pp 1112 - 1113; DOI: 10.1021/jm00293a022 |
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New thio derivatives of carcinogenic arylamines. 5. Ring-substituted methylthio-4-acetamidostilbenes T. Lloyd Fletcher, Moses J. Namkung, Hsi-Lung Pan, and Carol A. Cole pp 1113 - 1115; DOI: 10.1021/jm00293a023 |
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Antitumor activities and rates of hydrolysis of Schiff bases Ernest M. Hodnett and Joseph Tai pp 1115 - 1116; DOI: 10.1021/jm00293a024 |
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Potential antitumor agents. 1. Analogs of camptothecin J. A. Beisler pp 1116 - 1118; DOI: 10.1021/jm00293a025 |
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Gentamicin antibiotics. 4. Some condensation products of gentamicin C2 with aromatic and aliphatic aldehydes David J. Cooper, Jay Weinstein, and J. Allan Waitz pp 1118 - 1120; DOI: 10.1021/jm00293a026 |
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Catalytic hydrogenation of viomycin and capreomycin John R. Dyer, James H. Carter, and Pieter J. Van Wyk pp 1120 - 1121; DOI: 10.1021/jm00293a027 |
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Cobalt chelates of Schiff bases of aromatic amines as antitumor agents Ernest M. Hodnett, Charles H. Moore, and Frederic A. French pp 1121 - 1123; DOI: 10.1021/jm00293a028 |
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Synthesis and antifungal activity of substituted carbanilic acid esters I. Lalezari, H. Golgolab, and M. Emami pp 1123 - 1124; DOI: 10.1021/jm00293a029 |
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Absence of biochemical and pharmacological effects of the trypsinogen activation peptide John Kay, Beatrice Kassell, and Harris L. Friedman pp 1124 - 1126; DOI: 10.1021/jm00293a030 |
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Antimalarials. 8. 2,3-Trimethylene-4-quinoline amino alcohols. 5,7-Dichloro-2,3-dihydro-1H-cyclopenta[b]quinoline-9-(.alpha.-di-n-butylaminomethyl)methanol J. M. Sanders, D. P. Clifford, and R. E. Lutz pp 1126 - 1127; DOI: 10.1021/jm00293a031 |
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N,N1-.alpha.,.omega.-Alkylenebis(nitroacetamides) P. M. Carabateas pp 1127 - 1127; DOI: 10.1021/jm00293a032 |
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Tricyclic heterocycles derived from 4-oxo-4,5,6,7-tetrahydrothianaphthenes William A. Remers, Gabriel J. Gibs, John F. Poletto, and Martin J. Weiss pp 1127 - 1129; DOI: 10.1021/jm00293a033 |
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Synthesis and alkylation of tetrahydropyrrolo[3,4-c]pyrazoles Victor J. Bauer and S. R. Safir pp 1129 - 1130; DOI: 10.1021/jm00293a034 |
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Synthesis of some 5-substituted 10,11-dihydrodibenz[b,f]azepines R. W. Woodard, K. Baldzer, and D. W. Boykin pp 1131 - 1132; DOI: 10.1021/jm00293a035 |
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Analogs of amphetamine. 6. 2,5-Dimethoxy-4-methyl- and 2,5-dimethoxy-.alpha.,4-dimethylphenylalanines Beng T. Ho, L. Wayne Tansey, and Jen-Tzaw Huang pp 1132 - 1133; DOI: 10.1021/jm00293a036 |
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Synthesis of derivatives of N,N-dimethylhydrazine and their physiological activities W. Philip Brian pp 1133 - 1134; DOI: 10.1021/jm00293a037 |
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Comparisons of butyrylcholinesterase inhibitory potencies of selected 3-substituted-1-decylpiperidines with their electron charge densities O. Elmo Millner and William P. Purcell pp 1134 - 1136; DOI: 10.1021/jm00293a038 |
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Chemistry of cephalosporin antibiotics. 25. 3-Cyanomethyl cephem nucleus J. A. Webber and R. T. Vasileff pp 1136 - 1138; DOI: 10.1021/jm00293a039 |
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Synthesis and pharmacological activity of dialkylaminoalkyl esters of benzilic acids containing fluorine or trifluoromethyl groups I. Lalezari, M. Hatefi, M. A. Khoyi, N. Guiti, and F. Abtahi pp 1138 - 1140; DOI: 10.1021/jm00293a040 |
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Antineoplastic agents. XXVII. Single crystal x-ray structures of chemotherapeutic agents. 3. Structure of 1,4-diazabicyclo[2.2.1]heptanes, a new heterocyclic ring system Donald J. Abraham and Robert D. Rosenstein pp 1141 - 1142; DOI: 10.1021/jm00293a041 |
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Synthesis of enantiomeric chloroacetylcarnitine chlorides Ravindra C. Vasavada and Joseph G. Turcotte pp 1142 - 1142; DOI: 10.1021/jm00293a042 |
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3-Amino-4-hydroxy-L(-)-butyramide hydrochloride John C. Keresztesy, Arthur J. Zambito, and Robert D. Babson pp 1142 - 1143; DOI: 10.1021/jm00293a043 |
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Solid phase synthesis of [4-proline]oxytocin, [4-proline]mesotocin, [4-proline]glumitocin, and [4-lysine]mesotocin M. Manning, J. W. M. Baxter, T. C. Wuu, V. Smart-Abbey, K. Morton, E. J. Coy, and W. H. Sawyer pp 1143 - 1144; DOI: 10.1021/jm00293a044 |
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Book Reviews pp 1145 - 1146; DOI: 10.1021/jm00293a900 |
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Tumor inhibitors. 69. Structure-cytotoxicity relations among the sesquiterpene lactones S. Morris Kupchan, M. A. Eakin, and A. M. Thomas pp 1147 - 1152; DOI: 10.1021/jm00294a001 |
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Structure and tumor-promoting activity of anthralin (1,8-dihydroxy-9-anthrone) and related compounds Alvin Segal, Charline Katz, and Benjamin L. Van Duuren pp 1152 - 1154; DOI: 10.1021/jm00294a002 |
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Nucleoside peptides. 2. Synthesis of certain 5-N-aminoacyl and 5-N-peptidyl derivatives of 5-aminouridine George A. Ivanovics, Robert J. Rousseau, and Roland K. Robins pp 1155 - 1158; DOI: 10.1021/jm00294a003 |
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Nucleic acids. 11. Synthesis of 5'-esters of 1-.beta.-D-arabinofuranosylcytosine possessing antileukemic and immunosuppressive activity Duane T. Gish, Robert C. Kelly, Gerald W. Camiener, and William J. Wechter pp 1159 - 1162; DOI: 10.1021/jm00294a004 |
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Quantitative structure-activity relations in leucomycin and lincomycin antibiotics Yvonne C. Martin and Kathleen R. Lynn pp 1162 - 1166; DOI: 10.1021/jm00294a005 |
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Antimalarial agents. 8. Ring-substituted bis(4-aminophenyl) sulfones and their precursors Ivan C. Popoff, Allan R. Engle, Reginald L. Whitaker, and Gopal H. Singhal pp 1166 - 1169; DOI: 10.1021/jm00294a006 |
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Inhibition of electron transport by substituted salicyl-N-(n-octadecyl)amides Nivard Neft and Thomas M. Farley pp 1169 - 1170; DOI: 10.1021/jm00294a007 |
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Synthesis and antiinflammatory activity of some 3-carboxamides of 2-alkyl-4-hydroxy-2H-1,2-benzothiazine 1,1-dioxide Joseph G. Lombardino, Edward H. Wiseman, and W. M. McLamore pp 1171 - 1175; DOI: 10.1021/jm00294a008 |
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Excretion and metabolism of a nonsteroidal antiinflammatory agent, 4-hydroxy-2-methyl-2H-1,2-benzothiazine-3-carboxanilide 1,1-dioxide, in rat, dog, monkey, and man Josephine Chiaini, Edward H. Wiseman, and Joseph G. Lombardino pp 1175 - 1177; DOI: 10.1021/jm00294a009 |
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Metabolism of [14C]-verapamil Hugh M. McIlhenny pp 1178 - 1184; DOI: 10.1021/jm00294a010 |
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Potential antifertility agents. 1. Substituted diaryl derivatives of benzo[b]thiophenes, benzo[b]furans, 1H-2-benzothiapyrans, and 2H-1-benzothiapyrans R. R. Crenshaw, A. T. Jeffries, G. M. Luke, L. C. Cheney, and G. Bialy pp 1185 - 1190; DOI: 10.1021/jm00294a011 |
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17a-Propadienyl-19-nortestosterone and related compounds. New series of potent orally active progestogens M. Biollaz, R. M. Landeros, L. Cuellar, P. Crabbe, W. Rooks, J. A. Edwards, and J. H. Fried pp 1190 - 1192; DOI: 10.1021/jm00294a012 |
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1-Trifluoromethyl-1,2,2-triphenylethylenes. Synthesis and postcoital antifertility activity William J. Middleton, Diana Metzger, and Jack A. Snyder pp 1193 - 1197; DOI: 10.1021/jm00294a013 |
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Synthesis and hormonal activities of 8-L-homolysine-vasopressin Miklos Bodanszky and Gunnar Lindeberg pp 1197 - 1199; DOI: 10.1021/jm00294a014 |
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Thyroxine analogs. 21. o- and m-L-Thyroxine and related compounds Eugene C. Jorgensen and Peter E. Berteau pp 1199 - 1202; DOI: 10.1021/jm00294a015 |
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8-Substituted theophyllines. In vitro inhibition of 3',5'-cyclic adenosine monophosphate phosphodiesterase and pharmacological spectrum in mice Elizabeth B. Goodsell, Herman H. Stein, and Kathleen J. Wenzke pp 1202 - 1205; DOI: 10.1021/jm00294a016 |
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Linear free energy relations in the enzymic hydrolysis of substituted benzoylcholine esters James J. Zimmerman and Jere E. Goyan pp 1206 - 1211; DOI: 10.1021/jm00294a017 |
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Structure-activity relations having a basis in regular solution theory Arthur Cammarata, Suh Jen Yau, and Kenneth S. Rogers pp 1211 - 1212; DOI: 10.1021/jm00294a018 |
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Further evaluation of N,N'-polymethylene-bridged 2-aminoethanethiol derivatives and related compounds as radioprotective agents James R. Piper, Carl R. Stringfellow, and Thomas P. Johnston pp 1212 - 1217; DOI: 10.1021/jm00294a019 |
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2-Amino-5-nitroimidazoles Laird F. Miller and Ronald E. Bambury pp 1217 - 1218; DOI: 10.1021/jm00294a020 |
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Potential antimalarials. 6. 2-Phenyl-6- and -8-quinolinemethanols and 8-phenyl-4-quinolinemethanols J. B. Wommack, T. G. Barbee, K. N. Subbaswami, and D. E. Pearson pp 1218 - 1220; DOI: 10.1021/jm00294a021 |
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Potential antimalarials. 7. Tribromomethylquinolines and positive halogen compounds J. C. Craig and D. E. Pearson pp 1221 - 1222; DOI: 10.1021/jm00294a022 |
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Synthesis of some adamantane derivatives of 2-aminobenzothiazoles E. Costakis and P. Canonne pp 1222 - 1223; DOI: 10.1021/jm00294a023 |
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Antimicrobials. 1. Benzothiazolylbenzylamines P. J. Palmer, G. Hall, R. B. Trigg, and J. V. Warrington pp 1223 - 1225; DOI: 10.1021/jm00294a024 |
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Antimicrobials. 2. Substituted benzothiazolylbenzylamines and related compounds P. J. Palmer, R. J. Ward, and J. V. Warrington pp 1226 - 1227; DOI: 10.1021/jm00294a025 |
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Antimicrobials. 3. Benzothiazolylphenylalkylamines P. J. Palmer, R. B. Trigg, and J. V. Warrington pp 1228 - 1230; DOI: 10.1021/jm00294a026 |
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Synthesis and norepinephrine-depleting activity of some esters of metaraminol Walfred S. Saari, Andrew W. Raab, Charles S. Miller, William F. Hoffman, and Edward L. Engelhardt pp 1230 - 1233; DOI: 10.1021/jm00294a027 |
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Synthesis, transformation, and general pharmacologic activity in 1,4-benzodiazepine-3,5-diones Ned D. Heindel, William P. Fives, Thomas F. Lemke, Jay E. Rowe, Harry W. Snady, and Richard A. Carrano pp 1233 - 1235; DOI: 10.1021/jm00294a028 |
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Antispasmodic agents. 2. Syntheses and pharmacological activity of ethyl 2-(.omega.-aminoalkyl)-2-(3-methoxyphenyl)phenylacetates T. Kametani, K. Kigasawa, M. Hiragi, and T. Aoyama pp 1235 - 1237; DOI: 10.1021/jm00294a029 |
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Cholinergic receptor. 6. Synthesis and muscarinic activity of 2-methyl-4-(2-dimethylaminoethyl)-1,3-dioxolane methiodide K. J. Chang, H. F. Ridley, and D. J. Triggle pp 1237 - 1237; DOI: 10.1021/jm00294a030 |
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Potential folic acid antagonists. 5. Synthesis and dihydrofolate reductase inhibitory activities of 2-amino-4,6-substituted-5-arylazopyrimidines S. S. Chatterjee, S. Ludwig, J. F. Moran, D. J. Triggle, and A. Wayne pp 1237 - 1238; DOI: 10.1021/jm00294a031 |
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Antigenic polypeptides. Synthesis and immunochemical studies of poly(L-phenylalanyl-L-glutamyl-L-alanylglycyl)glycine-1-14C ethyl ester Brian J. Johnson and Charles Cheng pp 1238 - 1239; DOI: 10.1021/jm00294a032 |
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Synthesis and reactions of some pyrrolidinediones Jaysukhlal R. Merchant, Mehmood A. Hakim, Kutten S. Pillay, and Jimmy R. Patell pp 1239 - 1242; DOI: 10.1021/jm00294a033 |
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Preparation of some trimethylpentacyclo-[5.4.0.02,6.03,10.05,9]undecane-8,11-dione derivatives A. W. Chow, D. R. Jakas, and J. R. E. Hoover pp 1242 - 1243; DOI: 10.1021/jm00294a034 |
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Synthesis of thiocarbamate S-ester derivatives Robert J. Adamski, Satoru Numajiri, Richard Poe, Larry J. Spears, and Frederick C. Bach pp 1244 - 1244; DOI: 10.1021/jm00294a035 |
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Potential folic acid antagonists. 6. Potential irreversible folate reductase inhibitors derived from 2,4-diamino-5-arylazopyrimidines S. S. Chatterjee, J. F. Moran, D. J. Triggle, and A. Wayne pp 1244 - 1245; DOI: 10.1021/jm00294a036 |
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Pyrazoles. 4. Analogs of 3-(3,3-dimethyl-1-triazeno)pyrazole-4-carboxamide C. Wayne Noell and C. C. Cheng pp 1245 - 1246; DOI: 10.1021/jm00294a037 |
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Steroidal heterocycles. 14. 1,8a-Epoxy-1,4,4a,5,6,7,8,8a-octahydro-2-hydroxynaphthalene-3-carbonitrile and related compounds Helmut C. Neumann pp 1246 - 1246; DOI: 10.1021/jm00294a038 |
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Synthesis of 2-methylpteridine derivatives Sadao Nishigaki, K. Ogiwara, and Fumio Yoneda pp 1246 - 1247; DOI: 10.1021/jm00294a039 |
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A-Norandrogens Arvin P. Shroff and Robert B. Mason pp 1247 - 1247; DOI: 10.1021/jm00294a040 |
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Potential antineoplastics. 8. Synthesis and pharmacology of 6-methyl-2-thio-5-arylazouracils H. G. Garg and R. A. Sharma pp 1248 - 1248; DOI: 10.1021/jm00294a041 |
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Additions and Corrections - Choline Acetyltransferase Inhibitors. Configurational and Electronic Features of Styrylpyridine Analogs. C. J. Cavallito, H. S. Yun, J. C. Smith, and F. F. Foldes pp 1251 - 1251; DOI: 10.1021/jm00294a600 |
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Additions and Corrections - Azamorphinan and Related Compounds. III. Syntheses of 3-Hydroxy-N-substituted-9-azamorphinans. T. Kametani, K. Kigasawa, M. Hiiragi, N. Wagatsuma, K. Wakisaka, F. Satoh, and S. Saito pp 1251 - 1251; DOI: 10.1021/jm00294a601 |
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Additions and Corrections - Tranquilizing Drugs. Carbamates of 4-(4-Hydroxypiperidino)-4'-fluorobutyrophenone and Analogs. J. P. Li, R. G. Stein, J. H. Biel, J. A. Gylys, and S. A. Ridlon pp 1251 - 1251; DOI: 10.1021/jm00294a602 |
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Additions and Corrections - Synthesis and Activity of Some 3-Aryl- and 3-Aralkyl-1,2,3,4-tetrahydro-4-oxo-6-quinazolinesulfonamides. B. V. Shetty, L. A. Campanella, T. L. Thomas, M. Fedorchuk, T. A. Davidson, L. Michelson, H. Volz, S. E .Zimmerman, E. J. Belair, and A. P. Truant pp 1251 - 1251; DOI: 10.1021/jm00294a603 |
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Additions and Corrections - Synthesis and Pharmacology of N-Cyano-(β-arylethyl)amines. E. E. Smissman, A. C. Makriyannis, and E. J. Walaszek pp 1251 - 1251; DOI: 10.1021/jm00294a604 |
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Additions and Corrections - Potential Psychotomimetics. Bromomethoxyamphetamines. C. F .Barfknecht, and D. E. Nichols pp 1251 - 1251; DOI: 10.1021/jm00294a605 |
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Additions and Corrections - Interdependence between Physical Parameters and Selection of Substituent Groups for Correlation Studies. P. N . Craig pp 1251 - 1251; DOI: 10.1021/jm00294a606 |
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Additions and Corrections - Antimicrobial Compounds. 1. Synthesis and Antimicrobial Activity of Some Alkylidene, Cycloalkylidene, and Arylidene Derivatives of 3-Hydrazinopyridazine. M. Likar, B. Drinovec, M. Japelj, A. Pollak, A. Povse, and P. Jerman pp 1251 - 1251; DOI: 10.1021/jm00294a607 |
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Additions and Corrections - Prediction of the in Vitro Activity of Sulfonamides Synthesized from Simple Amines by Use of Electronic Data Obtained from the Simple Amines. J. K. Seydel pp 1251 - 1251; DOI: 10.1021/jm00294a608 |
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Additions and Corrections - A Conformational Study of Catecholamine Receptor Sites. 5. Syntheses of dl-3-Amino-2-(3,4-dihydroxyphenyl)-trans-2-decalol Hydrochlorides. E. Smissman, and R. T. Borchardt pp 1251 - 1251; DOI: 10.1021/jm00294a609 |
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Book Reviews pp 1249 - 1250; DOI: 10.1021/jm00294a900 |